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2-(2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
2-(2-hydroxyethyl)-8-(trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-{[(9-methyl-9H-carbazol-3-yl)formamido]methyl}-5-(pyridine-4-amido)benzoate
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(5-fluoro-2-methoxybenzoyl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
1-[(5-methylthiophen-2-yl)methyl]-2-(1,3-thiazol-2-yl)piperidine
ethyl 5-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-(4-fluorophenyl)-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperidine
1-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-indole-5-carboxamide
5-chloro-N-[(2,6-difluoro-3-methoxyphenyl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(4-methoxyphenyl)propan-1-one
methyl 3-(4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazol-1-yl)propanoate
3-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
5-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N3-tert-butyl-1-cyclohexyl-N5-[(2,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
7-[(4-fluorophenyl)methyl]-2-(3-methylbut-2-en-1-yl)-2,7-diazaspiro[4.5]decan-6-one
2-chloro-4-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-6-methoxyphenol
N-(carbamoylmethyl)-2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-chloro-4,6-dimethyl-3-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]benzene-1-sulfonamide
1-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
2-(4-ethylphenyl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
4-amino-2-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine-5-carbonitrile
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
N-benzyl-N-butyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-phenylpiperidin-4-amine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-(trifluoromethyl)-1H-pyrazole
2-amino-6-(2,4-dichlorophenyl)-4-(piperidin-3-yl)pyridine-3-carbonitrile
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[4-(trifluoromethyl)phenyl]urea
(3aR,6aR)-2-(3-ethoxypropanoyl)-5-(3-methylbut-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-1-propyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazole-4-carboxamide
4-{1-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
3-[1-(3-methoxy-5-methylthiophene-2-carbonyl)azetidin-3-yl]pyridine
2-(4-{[3-(2-methylphenyl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
N-methyl-6-oxo-N-[(4-phenoxyphenyl)methyl]piperidine-3-carboxamide
4-[(1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-cyclopropyl-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole