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N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(furan-2-ylmethyl)-2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]acetamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
{1-[2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]piperidin-2-yl}methanol
4-[(2R)-oxolane-2-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[methyl({4-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
4-(2-methyl-1H-imidazol-1-yl)-1-(pyridine-3-sulfonyl)piperidine-4-carboxylic acid
3-[methyl({2-methylthieno[2,3-d]pyrimidin-4-yl})amino]-1-phenylpropan-1-ol
2-[4-(hydroxymethyl)phenyl]-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3,4-dimethyl-5-sulfamoylbenzamide
6-(4-methoxyphenyl)-7-methyl-N-(oxan-3-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-ethyl-N-[(8-methoxy-2H-chromen-3-yl)methyl]oxan-4-amine
1-[4-(4-fluorophenyl)benzoyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
4-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)thiomorpholine
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]pyridine
2-(3-fluorophenyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)azepane-1-carboxamide
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(1H-imidazol-2-ylmethyl)-4-(oxan-4-yl)piperazine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2,4-difluoro-3-methoxybenzamide
(4aS,7aR)-1-[(2,5-dimethylphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(3-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
2-[(4aR,8aR)-4a-hydroxy-7-(6-methylpyridazin-3-yl)-decahydro-2,7-naphthyridin-2-yl]-N-cyclopropylacetamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
4-ethyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-{4-[2-(trifluoromethyl)morpholine-4-carbonyl]phenyl}ethan-1-amine
N-cyclopropyl-1-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2,2-dimethylpropanamide
2-amino-8-[3-(2-methylphenyl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-2-amine
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N-(propan-2-yl)-6-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidin-4-amine
4-methyl-N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
N-[2-(3-chlorophenyl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
9-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
3-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
2-{1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-2-yl}pyridine
3-[(3R,4S)-1-[6-(dimethylamino)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
methyl (2S,4S)-1-methyl-4-{6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-amido}pyrrolidine-2-carboxylate
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
1,5-dimethyl-4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(3S,4R)-N-(4-acetylphenyl)-3-(dimethylamino)-4-propylpyrrolidine-1-carboxamide
N-{[1-(1H-indol-3-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
[(1-methyl-1H-imidazol-2-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})propylamine