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3-[(3R,4S)-4-(dimethylamino)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]propan-1-ol
(3aS,7aR)-2-(2,3-dihydro-1H-inden-2-yl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-amino-4-(4,5-dimethylfuran-2-yl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
1-{2-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
1-(4-methoxyphenyl)-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-cyclopentyl-4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-oxobutanamide
8-(2,3-dihydro-1H-inden-2-yl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 4-{4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperazin-1-yl}benzoate
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}amino)-N-(1,3-thiazol-2-yl)propanamide
1-(1-benzofuran-2-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(2S,4S)-N-ethyl-4-(furan-3-amido)-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
N-butyl-N-cycloheptyl-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
N-[(1-benzylpiperidin-4-yl)methyl]-2-(4-hydroxypiperidin-1-yl)-N-methylacetamide
7-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(3-ethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,2S,9R)-11-[3-(3-hydroxy-3-methylbutyl)benzoyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
(1S,5R)-3-[2-(4-hydroxyphenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-(2-phenylethyl)piperazin-2-one
2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-6-methylquinolin-4-ol
2-cyclopropyl-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N,4-dimethylpyrimidine-5-carboxamide
5-[1-(piperidin-1-yl)ethyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]furan-2-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(4-fluorophenyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazin-2-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
(1S,6R)-9-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(4-chlorophenyl)-N-[2-methyl-5-(methylcarbamoyl)phenyl]morpholine-4-carboxamide
1-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
4-[({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1-cyclopropylpyrrolidin-2-one
4-(6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazine-2-carbonyl)morpholine
1-methyl-4-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(5-chloro-1H-indol-2-yl)methyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
(3R,4S)-N,N-dimethyl-1-(piperidine-1-sulfonyl)-4-(propan-2-yl)pyrrolidin-3-amine
3-(3-methylpyrazin-2-yl)-4H-chromen-4-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3,5-dimethoxybenzamide
2-(4-acetylpiperazin-1-yl)-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}acetic acid
4-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-phenoxy-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-(2,5-dimethylfuran-3-yl)-N,N-dimethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-[(3-methoxyphenyl)methyl]morpholine
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
N,2-dicyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}acetamide
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(oxolane-2-carbonyl)-decahydro-1,6-naphthyridine
1-[2-methoxy-5-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-methoxy-3-methyl-1H-indole-2-carboxamide