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ethyl 2-[4-(adamantan-1-yl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
8-fluoro-2-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
1-{4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-[(cyclopropylmethyl)sulfamoyl]-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methylbenzamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
8-[2-(methylamino)-2-phenylacetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-2-methanesulfonamido-N-[(5-methylthiophen-2-yl)methyl]propanamide
9-{2-[(3-methoxyphenyl)amino]butanoyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridine-2-carbonitrile
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-2,1-benzoxazole-3-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-methoxy-N-[3-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
1-(4-{[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-5-(4-methoxyphenyl)-1,2,4-triazine
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
2-ethyl-6-methyl-3-(4-phenylazepane-1-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridin-4-one
2-cyclopropyl-6-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
ethyl 2-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}-1,3-oxazole-4-carboxylate
N-(2-methoxyethyl)-N-{[2-(2-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}furan-2-carboxamide
N-[(3R,4S)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxyacetamide
N-[2-(2-ethylphenoxy)ethyl]-N-methylimidazo[1,2-a]pyridine-6-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
4-(propan-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-thiazole-2-carboxamide
N-[4-(3,3-diphenylpiperidin-1-yl)-4-oxobutyl]acetamide
methyl 4-[4-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
3-{[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
(1S,5R)-3-{imidazo[1,2-a]pyrimidine-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(prop-2-en-1-ylsulfanyl)propanamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]piperidin-4-amine
2-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-azaspiro[4.4]nonane
N-benzyl-3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carboxamide
[(3R,4R)-1-(8-chloroquinolin-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N2-methyl-N2-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidine-1,2-dicarboxamide
N-[3-(methylsulfanyl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-(5-{1-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
N-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
6-methoxy-N,3-dimethyl-N-(quinoxalin-6-ylmethyl)-1-benzofuran-2-carboxamide
N-(oxolan-3-ylmethyl)-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
methyl 6-(1-phenylcyclopropanecarbonyl)-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-ethyl-3-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}quinoline
N-({1-[(3-ethenylphenyl)methyl]pyrrolidin-3-yl}methyl)piperidine-4-carboxamide
3-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-(1-phenylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate