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methyl 2-(4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-2-oxopiperazin-1-yl)acetate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(2-methylpyrrolidin-1-yl)methyl]-N-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)benzamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-1-(1-benzofuran-5-ylmethyl)-N-ethyl-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
8-[2-(1H-imidazol-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-phenyl-1,2-oxazole-5-carboxamide
N,2-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3S,5R)-N3-(2-acetamidoethyl)-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
3-({2-[(3S)-3-ethylmorpholin-4-yl]acetamido}methyl)-4-methylbenzoic acid
2-methyl-6-(propan-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrimidin-4-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(pentan-3-yl)acetamide
4-[(2,5-difluorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]benzamide
N-(3-methoxypropyl)-1-methyl-N-(quinolin-5-ylmethyl)piperidin-4-amine
3-(4-hydroxyphenyl)-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-pyrazole-5-carboxamide
(3S,4S)-3-{[1-(3-chloro-4-methylphenyl)piperidin-4-yl](methyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
1-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperidine-4-carbonitrile
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-[1-(propan-2-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(pyridin-2-yl)-5-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-methyl-5-[2-(2,3,4-trimethoxyphenyl)phenyl]-1,3,4-thiadiazole
({[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}sulfamoyl)dimethylamine
(4aS,8aR)-6-[2-(dimethylamino)acetyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(propane-1-sulfonyl)piperidine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-cyclopropyl-1-{[4-(methylsulfanyl)phenyl]methyl}urea
N,1-dimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-indole-2-carboxamide
2-[1-(furan-2-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-yl]ethan-1-ol
(1s,4s)-4-[2-(naphthalen-1-yl)-1H-imidazol-1-yl]cyclohexan-1-amine
(2S,4S)-N-ethyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
1-{3-cyclopropyl-5-[2-(ethanesulfinyl)ethyl]-1H-1,2,4-triazol-1-yl}isoquinoline
2-({2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
(3R,4S)-4-cyclopropyl-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
4-(3-hydroxy-3-methylbutyl)-N-{2-[methyl(phenyl)amino]propyl}benzamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-amino-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-benzothiazole-5-carboxamide
1-(4-{[3-(1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-methoxyethan-1-one
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(oxan-3-ylmethyl)pyrimidin-2-amine
1-[cyclohexyl(methyl)amino]-3-{2-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
3-{[(2-hydroxyethyl)(methyl)amino]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
[1-(1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
8-[4-(aminomethyl)cyclohexanecarbonyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[5-(1H-indazol-1-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
4-(3-methylbutyl)-11-(morpholin-4-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[4-(difluoromethoxy)phenyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-[(2-chlorophenyl)methyl]-4-(morpholine-4-sulfonyl)morpholine
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(methylamino)ethan-1-one