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N-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
N-cyclopropyl-4-(3-hydroxy-3-methylbutyl)-N-(1H-indol-5-ylmethyl)benzamide
[(2,6-difluorophenyl)methyl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
5-[6-(piperazin-1-yl)pyridin-2-yl]thiophene-2-carbonitrile
4-[(4-carbamoylphenyl)methyl]-6-hydroxy-N,N-dimethyl-1,4-diazepane-1-carboxamide
(3R,9aR)-3-(2-methylpropyl)-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-[3-(2-fluorophenyl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-[2-(methylsulfanyl)pyrimidin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2,3-dihydro-1-benzofuran-7-carboxamide
5-cyclopropyl-1-(2-methoxyphenyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
4-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
2-methyl-4-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)-6-(pyrrolidin-1-yl)pyrimidine
3-{5-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
(2R,6S)-4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-2,6-dimethylmorpholine
5-{2-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
2-(2-chloro-4-fluorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
3-(2-oxopiperidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propyl-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
(3S,5S)-N-[(4-chlorophenyl)methyl]-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-(naphthalen-2-ylmethyl)pyrrolidin-3-amine
1-methyl-4-({5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,4-diazepane
5-(2,6-difluorophenoxymethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
4-phenyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine-4-carbonitrile
{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-cyclopentanecarbonyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-ethyl-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-(pyrrolidin-3-ylmethyl)-1,2-oxazole-3-carboxamide
(3S,4S)-4-cyclopropyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)pyrrolidine-3-carboxylic acid
N,8-dimethyl-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H-1,2,4-triazole-5-carboxamide
N,8-dimethyl-N-(2-phenylethyl)-3-[({[1-(propan-2-yl)pyrrolidin-3-yl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(3S,4R)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
ethyl 1-(3-{[(1-ethylpyrrolidin-2-yl)methyl]carbamoyl}-6-(4-methylthiophen-2-yl)pyridin-2-yl)piperidine-4-carboxylate
5-{5-[1-(furan-2-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(2-methyl-1-benzofuran-7-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
{1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]pyrrolidin-3-yl}methanamine
9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
methyl 4-[({1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)methyl]benzoate
N-[2-(furan-2-yl)ethyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{5-[2-(2-fluorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}pyrimidine
1-(4-phenylpiperazin-1-yl)-3-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}propan-1-one
2-{[(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[2-(4-fluorophenyl)ethyl]acetamide
1-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-4-phenylbutane-1,4-dione
N-methyl-2-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)acetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(furan-2-ylmethyl)piperidin-3-yl]propanamide