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2-benzyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3-thiazole-4-carboxamide
2-phenoxy-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(1-cycloheptylpiperidin-3-yl)-1-(3-methoxyphenyl)urea
3-(2,3-dihydro-1,4-benzodioxin-2-yl)-5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(propan-2-yl)-1,2,4-oxadiazole
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
(1S,3R)-3-amino-N-(2,1,3-benzoxadiazol-5-ylmethyl)cyclopentane-1-carboxamide
7-(2,5-dimethoxybenzenesulfonyl)-2-methyl-2,7-diazaspiro[4.5]decane
4-(2H-1,3-benzodioxole-5-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
1-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
(2S)-2-{2-[2-methoxy-5-(propan-2-yl)phenyl]-1H-imidazol-1-yl}-3-methylbutanamide
3-chloro-N-cyclopentyl-4-{[1-(3-hydroxypropyl)piperidin-4-yl]oxy}benzamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(propan-2-yl)piperazine-1-carbonyl]piperidin-2-one
N,N-diethyl-1-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-oxo-4H-chromene-2-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
N-({1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxyacetamide
1-[2-(2-methoxy-2-phenylacetamido)ethyl]-N-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
4-(5-ethyl-2-methylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(4aR,7aS)-4-[(2-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)-N-methylpyrimidin-2-amine
3-(5-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}acetamide
1-(4-acetylphenyl)-3-(thiolan-3-yl)urea
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(thiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[({1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
5-[(dimethyl-1,3-thiazol-4-yl)methyl]-3-methyl-1H-1,2,4-triazole
N-(1-methoxypropan-2-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[2-({7-methylpyrazolo[1,5-a]pyrimidin-6-yl}formamido)ethyl]piperidine-3-carboxamide
8-cyclopropanecarbonyl-2-[(4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2R,3R,6R)-3-phenyl-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2,5-dimethyl-3-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
2-ethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrimidine-5-carboxamide
5-ethyl-N,2-dimethyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrimidin-4-amine
2-(4,6-dimethylpyridin-3-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1H-imidazole
6-[4-(methylamino)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
(3S,5S)-1-(2,2-dimethylpropyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
1-(2-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-[(2R,4R,6S)-2-(3-hydroxyphenyl)-6-[2-(propylamino)pyrimidin-5-yl]oxan-4-yl]acetamide
1-[(3-ethoxyphenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
6-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
(4aS,8aS)-2-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-decahydroisoquinolin-4a-ol
4-[1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)piperidin-3-yl]benzoic acid
3-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,9-diazaspiro[5.5]undecane