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2-(2-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenoxy)ethan-1-ol
1-(4-chlorophenyl)-N-{[1-(1-methylpiperidine-4-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-{2-[(3-hydroxypiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
3,5-difluoro-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}benzamide
dimethyl({2-[2-(pyridin-4-yl)phenoxy]ethyl})amine
1,5-dimethyl-3-{[2-(thiophen-2-yl)-1H-imidazol-1-yl]methyl}-1H-indazole
8-(2,6-difluoro-4-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-fluoro-N-(4-{4-[(3-hydroxyadamantan-1-yl)amino]piperidin-1-yl}phenyl)benzamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(benzyl)amine
[3-(2,6-dimethoxyphenyl)-1H-1,2,4-triazol-5-yl]methanol
5-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-({2-[(3-cyano-2-methoxypyridin-4-yl)oxy]hex-5-en-1-yl}(methyl)amino)-N,N-dimethylacetamide
3-chloro-N-(2-methoxyethyl)-4-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}benzamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)acetamide
1-(carbamoylmethyl)-N-methyl-N-[(4-phenoxyphenyl)methyl]piperidine-4-carboxamide
N-(furan-2-ylmethyl)-5-{[(3-methoxyphenyl)methyl](methyl)amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1H-1,3-benzodiazole-5-carboxamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decane
5-(3-methoxyphenyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-1,2,4-triazin-3-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
ethyl 1-(2,6-dimethylpyrimidine-4-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(3-methylphenyl)piperidin-4-yl]acetamide
1-(2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrimidin-4-yl)piperidin-3-ol
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
N,1,4,6-tetramethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
{[3-(azonane-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl}diethylamine
N-[2-(dimethylamino)ethyl]-1-[1-(2,2-diphenylacetyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-phenyl-1,4-diazepane
2-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
methyl 5-[(butan-2-yl)amino]-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
5-tert-butyl-N-{3-[cyclopentyl(methyl)amino]propyl}-1,3,4-oxadiazol-2-amine
(1S,5R)-3-[2-hydroxy-3,5-bis(propan-2-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-butyl-2-{4-[(dimethylamino)methyl]phenyl}-3,4-dihydropyrimidin-4-one
N-[(2-ethylpyrimidin-4-yl)methyl]-N-methylthian-4-amine
1-(azocan-1-yl)-3-[5-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
6-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1,4-oxazepan-6-ol
2-(1H-imidazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
6-fluoro-3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinolin-4-ol
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3-(1H-pyrazol-5-yl)piperidine
N-{1-[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]propan-2-yl}-2-methylbenzamide
1-{2-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methylpiperazine
N-ethyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(2-methylprop-2-en-1-yl)benzamide
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine-1-carboxamide
2-(cyclopropylmethyl)-7-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one