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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
5-acetyl-N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{spiro[2.5]octan-1-ylmethyl}piperazine
N-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
4-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]pyridine
{[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}oxane-2-carboxamide
(3R,5S)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(cyclopropylmethyl)-7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}ethan-1-one
6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-cyclobutyl-3-methyl-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-ol
4-cyclobutaneamido-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}benzamide
N-(4-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
2-methyl-1-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}azetidin-3-yl)piperidine
N-[(2-methoxynaphthalen-1-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[2-(2-methylpropanesulfonyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
5-fluoro-N2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-N4,N4-dimethylpyrimidine-2,4-diamine
5-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-[3-(furan-2-yl)phenyl]-N-(oxan-4-ylmethyl)piperidin-4-amine
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N-cyclohexyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-(2,2-dimethyloxan-4-yl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(5-methylpyridin-2-yl)ethyl]benzamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
3-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}benzonitrile
4-(1H-imidazol-1-yl)-1-[3-(5-methylfuran-2-yl)butyl]piperidine-4-carboxylic acid
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-{[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-(3-methoxypropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
(2S)-2-amino-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-4-(methylsulfanyl)butanamide
2-(4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]oxane-4-carboxamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
4-({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
N-[(3S,4R)-1-(1-benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
dimethyl[2-(4-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-1-yl)ethyl]amine
6-[({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-methyl-5-[3-(pyridin-4-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[5-(1H-indol-5-yl)-2-methoxyphenyl]methyl}(methyl)amine
8-(4-methoxy-3-methylbenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2-chlorophenyl)methyl]-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
2-(1H-pyrazol-1-yl)-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethan-1-one
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N-[(2-methoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-butyl-N-(pyridin-2-ylmethyl)quinoxaline-5-carboxamide