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N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-ethoxyphenol
N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(2-methoxyphenyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazole-4-carboxamide
N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(cyclopropylcarbamoyl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-benzyl-3-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
6-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1H-indole
2-{2-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethan-1-ol
7-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-1-(1,2-oxazol-3-ylmethyl)-N-(2-phenylethyl)piperidin-3-amine
3,4-dimethyl-N-(prop-2-en-1-yl)-N-(propan-2-yl)-5-sulfamoylbenzamide
2-{4-[3-(1,2-oxazinan-2-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[1-(2,5-difluorophenyl)cyclopropyl]-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
(2R,3R,6R)-3-(4-fluorophenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-{[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}phenyl)imidazolidin-2-one
2-[4-(2-ethylphenyl)piperazin-1-yl]-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
methyl 4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}benzoate
N-[2-methoxy-4-(pyrimidin-5-yl)phenyl]acetamide
(3S,9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidin-4-yl}methanesulfonamide
N6-(2-methoxyethyl)-N5-methyl-N5-[(1-methylpiperidin-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-amino-3-ethyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(3-phenoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[4-(1H-indol-3-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
2-(3-fluorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
6-[6-(dimethylamino)pyridine-3-carbonyl]-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
6-methyl-N-(1,3-thiazol-2-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-{4-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
6-(3,4-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,2,4-triazole-5-carboxamide
1-(quinoxalin-2-yl)azepan-4-amine
1-tert-butyl-N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-5-oxopyrrolidine-3-carboxamide
(1S,2R)-N2-butyl-N1-methyl-N1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]cyclohexane-1,2-dicarboxamide
2-{3-[1-(dimethylamino)ethyl]phenyl}-6,7-dimethoxyquinazolin-4-amine
methyl 3-acetamido-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
4-[(4-fluorophenyl)methyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(1R,2S)-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-propylcyclopropane-1-carboxamide
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
3-[(2,6-dimethoxyphenyl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-butyl-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
5-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-2-hydroxybenzoic acid
1-(4-chlorophenyl)-N-{[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide