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3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
4-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-1λ6-thiomorpholine-1,1-dione
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]acetamide
3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-5-(trifluoromethyl)-1H-1,2,4-triazole
4-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-4-(1,2,4-oxadiazol-3-yl)piperidine
2-[2-(butan-2-yl)phenoxy]-N-cyclopropyl-N-(pyridin-3-ylmethyl)acetamide
4-{3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[2-(propan-2-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-4-hydroxyphenyl)acetamide
2-butyl-8-(2,4-difluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}pyrimidine-5-carboxylic acid
1-(pyridin-2-yl)-4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperazine
3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-methyl-1H-imidazol-1-yl)acetamide
4-[3-(1-benzothiophen-2-yl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
2-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-fluoro-N-(1-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
6-methyl-2-({[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)quinolin-4-ol
N-({7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
methyl 8-(1,3-benzothiazol-2-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
(1R,2S,6R,7S)-4-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}-4-azatricyclo[5.2.2.02,6]undecane
2-({[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}amino)-N-(1,3-thiazol-2-yl)propanamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)-2-(1,3-thiazol-2-yl)piperidine
1-[1'-(6-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-[5-(2-amino-1,3-benzothiazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-{2-[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}pyrrolidin-2-one
(1R,3S)-7-(4-hydroxy-3-methoxybenzoyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
N-propyl-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
2-(3,4,5-trimethoxyphenyl)-1,3-thiazole-4-carboxamide
1-(4-methylpent-3-en-1-yl)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(4aS,7aR)-1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclohexyl-N-(pyridin-4-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
6-methoxy-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[(2,5-difluorophenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
(3R,4S)-1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-3,4-dimethylpiperidin-4-ol
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(morpholine-4-sulfonyl)benzamide
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
2-{9-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
1-ethyl-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-(pyridin-2-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-1-[(4-methylphenyl)amino]-N-[3-(oxolan-2-yl)propyl]cyclopentane-1-carboxamide
(3S,4S)-4-[4-(cyclopentylmethyl)piperazin-1-yl]-1-(4-methoxybenzoyl)pyrrolidin-3-ol
4-ethyl-3-(piperidin-3-yl)-1-(2-propoxyethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one