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1-(2-methylquinolin-5-yl)-3-(thiolan-3-yl)urea
N-ethyl-2-(4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)acetamide
methyl (2R,4S)-4-hydroxy-1-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]piperidine-2-carboxylate
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yl)propyl]amine
3-ethyl-5-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1,2-oxazole-4-carboxamide
1-{2-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-hydroxypropan-1-one
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})methylamine
4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-oxazepan-6-ol
2-{1-tert-butyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
(2R,6S)-4-(5-{[4-(3-methoxypropyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-2,6-dimethylmorpholine
1-cyclopentyl-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2-methyl-8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(dimethylamino)-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-(4-methylphenyl)ethan-1-one
2-ethyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-cyclopropyl-2-fluoro-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}benzamide
4,6-dimethoxy-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}propanamide
9-methoxy-3-[(4-oxo-4H-chromen-3-yl)methyl]-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-methoxy-N-[(6-methylpyridin-2-yl)methyl]benzamide
3-(1-butyl-1H-imidazol-2-yl)-N-(2,4-dimethoxyphenyl)piperidine-1-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
2-(3-propylmorpholine-4-carbonyl)-4H-chromen-4-one
4-[(methylsulfanyl)methyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
2-amino-4-(2-butyl-1H-imidazol-4-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-({1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}methyl)-4-fluorobenzamide
7-{2-[(3,5-dimethylphenyl)carbamoyl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(3-{2-[2-(methoxymethyl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)-1H-1,3-benzodiazole
4-acetyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
1-(2-methoxyethyl)-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
(1S,5R)-6-(2-methoxyethyl)-3-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[(2-fluorophenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
6-[4-(2-methoxyethoxy)phenyl]quinoline
methyl 5-{[(3-hydroxyphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{2-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(2,3-dimethylphenyl)-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1-propyl-1H-pyrazole-4-carboxamide
N-(2,3-dihydro-1H-inden-4-yl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
5-{1-[2-(6-methyl-1-benzofuran-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(benzyloxy)-1-(furan-2-ylmethyl)piperidine
2-{5-[2-(morpholin-4-yl)ethyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-ethyl-N-(2-methoxyethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-N-methyloxolan-3-amine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-(4-methylphenyl)propanamide
7-(cyclopropylmethyl)-2-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
{[5-(3-chlorophenyl)furan-2-yl]methyl}(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine