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1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(methoxymethyl)piperidine
(3R)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(3-propyl-1H-pyrazole-5-carbonyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methoxybenzoyl)piperazine
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-(3,4-dimethoxyphenyl)ethan-1-one
2-methoxy-N-[3-({[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
6-(2-aminoethyl)-2-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
3-[1-(isoquinoline-3-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
2-(1-butyl-1H-pyrazol-4-yl)-7-chloro-N,N-dimethylquinoline-4-carboxamide
N-{[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenylacetamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
2-methyl-6-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}pyrimidin-4-ol
2-ethyl-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidine-5-carboxamide
1-(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}piperidin-1-yl)ethan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3,6-dimethylpyrazin-2-yl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amine
N-[1-(2-methylphenyl)cyclopropyl]-3-(1-methylpiperidin-2-yl)propanamide
(4aS,7aR)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1H-indazol-3-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
2-{5-[6-(morpholin-4-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-(dimethylamino)-2-(3-methylphenyl)-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)acetamide
N-(2-methoxyethyl)-4-methyl-3-[(propylcarbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(2-methoxyethyl)-5,6-dimethyl-N-(1-methylpiperidin-4-yl)pyridine-3-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
(1S,5R)-6-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
4-(benzylamino)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}butan-1-one
N-{4-[(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenyl}acetamide
N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1-(pyridin-2-yl)piperidine-3-carboxamide
(4aS,8aR)-6-(1-benzofuran-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-{3-methyl-5-[(4-oxo-3,4-dihydroquinazolin-3-yl)methyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(4aR,7aS)-4-[(4-chlorophenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{1-benzyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(5S)-5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-(3-methoxyphenyl)piperidine-1-carboxamide
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-cyclopentyl-1,4-diazepane
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-2-methyl-4-phenylpiperazine
N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-{2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
N-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
3-(2-cyclopropylphenyl)-1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
1-ethyl-8-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione