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3-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-(5-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
N-[(3-chlorophenyl)methyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-(2-aminoethyl)-N-methyl-N-(2-phenylethyl)pyrimidin-4-amine
N-{3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}cyclopropanecarboxamide
2-(1,3-thiazol-4-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
(1-{[1-(5-methyl-2-phenylfuran-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
4-ethyl-3-(1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2-ethylpyrimidine-5-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2,4-dimethoxybenzoyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
5-{6-methylimidazo[1,2-a]pyridin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-({[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
5-fluoro-N,N-dimethyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-benzyl-9-{thieno[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
ethyl 3-benzyl-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine-3-carboxylate
methyl 7-oxo-3-(3-phenylprop-2-ynoyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-benzyl-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-sulfonamide
N-(3-ethoxypropyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)quinoline-3-carboxamide
(1S,5R)-3-(4-methylbenzoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-2-[1-(1H-indazole-3-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
2-{4-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carboxamide
6-(propan-2-yl)-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
N-[2-(pyridin-2-yl)ethyl]-6-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-[(3R,4S)-1-(3-fluoropyridin-2-yl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
1-[(2,4-difluorophenyl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-[4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-3,5-dimethyl-1H-pyrazol-1-yl]ethan-1-ol
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(2,5-dimethylfuran-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R,6R)-10-methoxy-4-[2-(morpholin-4-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[2-(2-chlorophenyl)ethyl]-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(dimethylamino)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-[2-(dimethylamino)ethyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
4-methyl-6-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-2-(pyridin-3-yl)pyrimidine
(1R,5R)-N,N-dimethyl-6-(quinolin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
5-ethyl-5-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4-propylpyrimidine-5-carboxamide
N-[4-(4-acetyl-6-hydroxy-1,4-diazepane-1-carbonyl)phenyl]ethane-1-sulfonamide
N-[(1R)-1-phenylethyl]-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-methyl-8-(1,3,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(4-{[(benzylsulfamoyl)amino]methyl}oxan-4-yl)methanol
N-(2,4-dimethylphenyl)-3-[(2-ethylpyrimidin-5-yl)formamido]propanamide
13-(2-propoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
5,6-dimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyridine-3-carboxamide
3-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-N-(pyridin-3-ylmethyl)formamido}propanoic acid