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3-(2-methoxyphenoxymethyl)-5-[1-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazole
2,3-dimethyl-6-(2,7,8-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[(3-ethoxy-4-methoxyphenyl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(4-cyclopentylpiperazin-1-yl)-2-(2,3-dimethoxy-5-methylphenyl)acetic acid
4-({1-[(2R)-2-aminopropanoyl]piperidin-4-yl}oxy)-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
4-ethyl-5-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
(3S)-4-[3-(difluoromethoxy)benzoyl]-3-ethylmorpholine
N4-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
(3aS,6aS)-2-acetyl-5-[5-(dimethylcarbamoyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[5-(3-methyl-1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
3-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
4-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}pyrimidine-5-carboxylic acid
7-[(3-methoxyphenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
6-(2-fluoro-6-methoxyphenyl)-1,2,3,4-tetrahydroquinazoline-2,4-dione
2-ethoxy-6-[(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amine
methyl 3-[7-chloro-2-(propanamidomethyl)-2,3-dihydro-1-benzofuran-5-yl]benzoate
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
9-(cyclopropylmethyl)-1-methyl-4-(1,3-thiazol-4-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethoxy]ethan-1-ol
methyl 2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(2-methoxyphenyl)ethyl]propanamide
3-{1-[2-(pyridin-2-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2H-1,3-benzodioxole-5-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)pyridine-3-sulfonamide
N-[(3S,4R)-1-[3-(3-fluorophenyl)propanoyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
6-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-2-methylpyrimidin-4-ol
propyl N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
ethyl 2-[(5-{[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]methyl}pyrimidin-2-yl)(methyl)amino]acetate
[(2,3-difluorophenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-(4-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
ethyl 3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}butanoate
2-(methylamino)-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
5-[(methylsulfanyl)methyl]-N-[2-(pyrrolidine-1-sulfonyl)ethyl]furan-2-carboxamide
N-(3,3-diphenylpropyl)-6-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
6-(2,4-dimethoxyphenyl)-N2,N2-diethylpyrimidine-2,4-diamine
5-[6-(methoxymethyl)pyrimidin-4-yl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(2,6-difluorophenoxymethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methylpyrimidin-4-amine
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(5-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazole