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N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}-5-methoxyfuran-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,3-oxazole-4-carboxamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]pyrimidin-2-amine
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(4-methoxyphenoxymethyl)piperidine
(3aR,6aR)-2-methanesulfonyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(adamantan-1-yl)-4-hydroxy-N-(1,2-oxazol-3-ylmethyl)pyrimidine-5-carboxamide
1,2-dimethyl-5-{[2-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}-1H-1,3-benzodiazole
6-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
6-methyl-2-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxylic acid
N-[(3R,4R)-1-[(2,4-difluorophenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(phenylsulfanyl)ethan-1-one
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(cyclohexylsulfanyl)propyl]-3-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
7-chloro-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-9H-fluoren-9-one
1-[4-(1-benzofuran-2-ylmethyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-4-phenylpiperazine
N,1-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-indole-3-carboxamide
N-[(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
(2E)-N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide
4-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-2-(1H-pyrazol-3-yl)pyridine
N-(2,2-diphenylethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-[2-(2-fluorophenoxy)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(3R,9aR)-3-(2-methylpropyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
N-cycloheptyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
2-(methylsulfanyl)-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyrimidine
3-(1H-imidazol-4-ylmethyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
4-{5-[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-yl}morpholine
(2R,6S)-4-{[5-(5-fluoropyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,6-dimethylmorpholine
2-{1-cyclohexyl-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1'-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(piperidin-2-yl)ethyl]-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(1S,4S)-2-(2-chlorophenyl)-5-(3,5-dimethoxybenzoyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N,1-dimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-[4-(3-cyanopiperidin-1-yl)-2-(dimethylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetic acid
3-benzyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,5R)-3-(2,3,6-trimethylquinoline-4-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,2,5,7-tetramethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
6-(3-fluorophenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(cyclobutylmethyl)-1-(4-fluoro-3-methoxyphenyl)-3-(oxolan-2-ylmethyl)urea
(2R,3R,6R)-3-phenyl-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(pyridin-3-ylmethyl)-4-(quinolin-6-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
1'-(4,6-dimethylpyrimidin-2-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]