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naphthalen-1-yl (7S,9aR)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
2-[benzyl(pyridin-2-ylmethyl)amino]-2-methylpropan-1-ol
8-(2-phenylquinazolin-4-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-(methoxymethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[(4-acetamidophenyl)methyl]-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
7-(cyclobutylmethyl)-2-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-tert-butyl-4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]pyrrolidin-2-one
3-methoxy-5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
{5-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]furan-2-yl}methanol
ethyl 4-(cyclopropylmethyl)-1-[(5-ethylfuran-2-yl)methyl]piperidine-4-carboxylate
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-(2-chloroprop-2-en-1-yl)-3-({[(2-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
methyl 4-(5-{[(1-carbamoylethyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-(4-{[(4-methoxypyridin-2-yl)methyl]amino}-6-methylpyrimidin-2-yl)phenol
2-(dimethyl-1,3-thiazol-5-yl)-N,N-bis(propan-2-yl)benzamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
1-(4-methoxyphenyl)-6,6-dimethyl-N-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1R,9S)-5-amino-3-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-[3-methoxy-5-(trifluoromethyl)phenyl]-3-(2-methoxyethyl)-3-methylurea
ethyl 4-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine-4-carboxamide
1-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-(4-chloro-3-fluorobenzoyl)-4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
1-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-2-ol
4-({4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridin-2-ol
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
5-ethyl-N,2-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidin-4-amine
3-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
2-(5-methyl-1H-pyrazol-1-yl)-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
3-{5-[6-(hydroxymethyl)pyridine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
methyl 5-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-methyl-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}piperidine
(3S,9R)-11-(3-fluoro-4-methylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-methyl-4-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}piperidine
(2E)-3-(2,3-difluorophenyl)-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]prop-2-en-1-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-(4-methoxyphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]acetamide
3-({[5-methyl-6-(4-phenylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
4-(3-ethynylbenzoyl)-2-(2-phenylethyl)morpholine
{4-[(4-methoxyphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidin-4-yl}methanol
4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]morpholine
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(1H-1,3-benzodiazol-2-ylmethyl)-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane