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2-amino-N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-6-methylpyrimidine-4-carboxamide
3-acetamido-N-{1-[(4-methylphenyl)methyl]cyclopropyl}benzamide
1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-{2-oxo-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethyl}pyrrolidin-2-one
3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
2-{2-[2-(4-chlorophenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
3-[2-(4-fluorophenyl)ethyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
1-[(2-fluorophenyl)methoxy]-8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
2-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(1-hydroxyethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]-9H-purine
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazole-2-carboxamide
1-methyl-3-propyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
1-cyclopentyl-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidin-2-one
1-(3-{[4-(methoxymethyl)piperidin-1-yl]methyl}-6-methylquinolin-2-yl)piperidin-3-ol
2-(6-cyclopropylpyrimidin-4-yl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
2-methyl-5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]phenol
1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
N-(1-cyclopropanecarbonylpiperidin-3-yl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-benzyl-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine
2-({4-[1-(naphthalen-1-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)pyrimidine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-6-carboxylic acid
2-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1-[(4-methoxyphenyl)methyl]-1H-imidazole
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
2-(2-phenylethyl)-4-[1-(pyrazine-2-carbonyl)piperidin-4-yl]morpholine
4-[2-(benzyloxy)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-(4-methylpiperazine-1-carbonyl)pyridin-2-amine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidin-2-amine
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
3-{3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propoxy}pyridine
2-[3-(5-chlorothiophen-2-yl)-4-methyl-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
5-[3-(4-acetylpiperazin-1-yl)-3-oxopropyl]-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
2-amino-6-(furan-2-yl)-4-[4-methoxy-3-(methoxymethyl)phenyl]pyridine-3-carbonitrile
6-ethyl-N-[1-(thian-4-yl)piperidin-4-yl]pyrimidin-4-amine
N-methyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-N-(pyrazin-2-ylmethyl)piperidin-4-amine
(5-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}furan-2-yl)methanol
8-acetyl-2-(1-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}-3-phenylpropan-1-one
ethyl 2-{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-2-yl}acetate
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(2-phenoxyethyl)piperazine
1-cyclopentanecarbonyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidine-4-carboxamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}azocane
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrrol-1-yl)butan-1-one
10-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
3-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)furan-2-carboxamide
(1S,2S)-2-{4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl}cyclohexan-1-ol