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8-fluoro-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-2-carboxamide
methyl 5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
1-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 5-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cyclohexyl-N-methyl-2-phenylacetamide
(4aS,7aR)-1-(3-hydroxy-2-methylbenzoyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
(3E)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]hex-3-en-1-one
3-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-(2-benzamido-5-methylphenyl)-1H-1,2,4-triazole-5-carboxamide
1-{6-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyridin-3-yl}ethan-1-one
N-[4-(pyridin-2-ylmethoxy)phenyl]azocane-1-carboxamide
N-[(4-fluoro-3-methylphenyl)methyl]-3-(pyrrolidin-3-yl)benzamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(4-fluorophenoxy)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-benzoyl-6-(2-fluoro-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
3-({2-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[3-(2-methylphenyl)piperidin-1-yl]pyrimidine
5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(ethanesulfonyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
5-chloro-N-(2-methoxyethyl)-3-methyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
(2-{3-[3-(3-fluoropyridin-4-yl)phenyl]-1H-pyrazol-1-yl}ethyl)dimethylamine
2-(azepan-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-(3-carbamoyl-4-methoxyphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
5-[2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-fluoro-4-hydroxyphenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
dimethyl[2-(2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-N4,6-dimethylpyrimidine-2,4-diamine
(2S,4S)-4-amino-1-(3,5-difluoro-4-methoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
2-ethyl-4-methyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,3-oxazole-5-carboxamide
2-(2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
1-(5-fluoropyridin-3-yl)-3-(2-methanesulfonamidoethyl)urea
5-fluoro-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}quinazolin-4-amine
2-amino-6-(4-hydroxyphenyl)-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(3S,4S)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-(piperidin-1-yl)pyrrolidin-3-ol
1-{2-[4-(2-fluorophenoxy)piperidin-1-yl]ethyl}-1H-indazole
1-[(4-fluoro-2-methylphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-cyclopropanecarbonyl-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
(2-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}thiophene-3-sulfonamide
1-(2,6-dimethylpyridin-3-yl)-3-[(2S)-1-methoxypropan-2-yl]urea
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
(1R,5R)-3-methanesulfonyl-6-[(5-phenylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1R,7S)-3-(2,2-dimethylpropyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(furan-2-ylmethyl)acetamide