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1-(6-aminopyridine-3-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-({[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)piperidin-3-ol
1-(oxolan-2-ylmethyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-(2,4-dimethoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(2E)-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-2-yl)prop-2-enamide
N-cyclopropyl-1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]piperidine-3-carboxamide
[1-(4,6-dimethylpyrimidin-2-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
4-{1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}pyridine
3-({4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)benzonitrile
2-(3-methyl-1,2-oxazol-5-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
(2R,6R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-{2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetyl}piperidine-4-carbonitrile
1,3,7-trimethyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
2-{[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]amino}-N-(pyrazin-2-yl)acetamide
N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
2-[4-(1H-indole-2-carbonyl)morpholin-3-yl]-N-(4-methoxyphenyl)acetamide
methyl 4-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]carbamoyl}butanoate
1-cyclopentyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
[(3S,5R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-({[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
N-[2-(2-methoxyphenyl)-1-methyl-5-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl]acetamide
9-[(4-ethylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-(pyrrolidin-1-yl)benzamide
1-[2-(2,3-dimethoxyphenyl)ethyl]-2-(furan-2-yl)-1H-imidazole
2-[(cyclopropylmethyl)sulfanyl]-1-[(3S,4S)-3-hydroxy-4-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-1-yl]ethan-1-one
(1R,5R)-6-[2-(2-methoxyphenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(3-methoxyphenyl)methyl]urea
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)urea
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-ethyl-3-[(1-methyl-2-oxopyrrolidin-3-yl)sulfamoyl]-N-(2-methylprop-2-en-1-yl)benzamide
{1-[4-(hydroxymethyl)benzoyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
N,6-dimethyl-4-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[4-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)piperazin-1-yl]-N-ethylacetamide
[(4-fluorophenyl)methyl]({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
N2-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-N4-ethylpyrimidine-2,4-diamine
2-{4-[(4-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
7-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-[(adamantan-1-ylformamido)methyl]-5-(1,3-dimethyl-1H-pyrazole-5-amido)benzoate
1-methoxy-8-[(3-methylthiophen-2-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
1-(4-methoxyphenyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
[7-(pyridin-4-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methanamine
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole