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N-(2-fluorophenyl)-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
1-(6-chloro-2-methylpyridin-3-yl)-3-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]urea
2-methyl-4-(4-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}phenyl)butan-2-ol
(2S)-2,3-diamino-1-[2-(5,6-dichloro-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-[(thiophen-2-ylmethyl)carbamoyl]piperidine-4-carboxylic acid
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine-3-carboxylate
N-ethyl-2-(2-fluoro-5-methoxyphenyl)pyrimidin-4-amine
(2S,4S)-1-cyclohexyl-N-ethyl-4-[2-(3-hydroxyphenyl)acetamido]pyrrolidine-2-carboxamide
3-{3-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
(1R,6S)-9-methyl-N-(2-phenylethyl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
2-hydroxy-5-[1-(4-sulfamoylphenyl)-1H-imidazol-2-yl]benzoic acid
N-(cyclohex-1-en-1-ylmethyl)-6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S)-2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)-3-(4-hydroxyphenyl)propanamide
(4aS,8aS)-2-cyclohexyl-7-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-5-(4-fluorophenyl)-2H-1,2,3,4-tetrazole
4-[(4-methoxynaphthalen-1-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-phenylethyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(pyridin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
(3aR,6aR)-2-(2-methoxyethyl)-5-[2-(methylsulfanyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(3-hydroxy-3-methylbutyl)benzoyl]azepan-4-ol
(3aR,6aR)-2-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(cyclopropylmethyl)-7-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-acetyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}thiophene-2-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-1-ethyl-1H-1,2,4-triazol-3-yl}acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[2-({5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}amino)ethyl]acetamide
N5-[(6-methoxy-2H-chromen-3-yl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
7-(3-methyl-2-oxoimidazolidin-1-yl)-4-(3-methylthiophen-2-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-({1-[6-(1,4-diazepan-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-amino-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)acetamide
(4aR,8aR)-2-methanesulfonyl-7-(1-methyl-1H-pyrrole-2-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
N-[2-(2-fluorophenyl)-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
N-(2-{7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
(2S)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-2-carboxamide
1-methyl-1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-methyl-4-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-indole
9-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-acetyl-1H-pyrazol-1-yl)-N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
3-(4-hydroxyphenyl)-N-(2-oxoazepan-3-yl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazine-1-sulfonamide
4-[(2,6-difluoro-4-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-fluorophenyl)-N-(4-{4-[(oxan-4-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
(5S)-5-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
(3S,4R)-1-[3-(2-oxoazepan-1-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
N,N-dimethyl-6-(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carboxamide