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(2R,3S,6R)-3-phenyl-5-(quinoline-8-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aR)-6-(6-aminopyrimidin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(4-{[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}phenyl)acetamide
3-[(3-ethenylphenyl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
3-[(2-fluorophenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,5S)-5-{1-[(4-ethylphenyl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl}pyrrolidin-3-ol
[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
5-(1H-imidazol-1-ylmethyl)-2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
2-[2-methyl-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)-1H-indol-1-yl]acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
1-{4-[2-(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethoxy]phenyl}propan-1-one
1'-(7-methyl-1-benzofuran-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(1,2,3-thiadiazol-5-yl)urea
4-(4-methyl-1H-pyrazol-1-yl)-1-[(propan-2-yl)carbamoyl]piperidine-4-carboxylic acid
1-ethyl-3-(pyridin-2-ylmethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-methoxypyrimidin-4-amine
N-[1-(2-chlorophenyl)ethyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-methyl-4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-{ethyl[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]amino}-1λ6-thiolane-1,1-dione
{4-fluoro-7-[6-(propan-2-yl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
(3S,4S)-1-[(3-fluorophenyl)methyl]-4-[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]pyrrolidin-3-ol
({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
5-{5-[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
N-{5-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-yl}acetamide
(3S,4S)-4-(propan-2-yloxy)-1-(2,5,7-trimethylquinoline-4-carbonyl)pyrrolidin-3-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-imidazole-2-carboxamide
2-(2-methoxyethyl)-8-(5-propylthiophene-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-methoxyphenyl)-3-methyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
7-(3,5-dimethoxyphenyl)-1,2-dihydroisoquinolin-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-[1-(3,4-dimethylphenyl)-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-7-yl}-1H-1,2,4-triazol-3-yl]acetamide
2-[4-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
5-(3-phenylphenyl)pyrazin-2-amine
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(benzyloxy)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-methyl-1,3-benzoxazole-6-carbonyl)pyrrolidin-3-yl]methanol
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-1-methylpiperidine-2-carboxamide
4-[1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
4-(4-chlorophenyl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]butan-1-one
N-[(5-chlorothiophen-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
{4-[(dimethylamino)methyl]-1-[4-(2-fluorophenyl)benzoyl]piperidin-4-yl}methanol
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(morpholin-4-ylmethyl)-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,4-oxazepane
N,N,1-trimethyl-6-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-fluoro-N-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide