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N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-methyl-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-indole
11-acetyl-4-[(2,6-dimethoxyphenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
9-ethyl-1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(4-hydroxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(4aS,7aR)-1-(3-acetyl-1H-pyrazole-5-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(3-fluoro-4-methoxyphenyl)-3-[3-(methoxymethyl)pyrrolidin-1-yl]-1,2,4-triazine
2-{2-chloro-6-methoxy-4-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}acetamide
(3-{2-[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethyl)piperidin-3-ol
1-[6-methyl-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
1-[(3-fluorophenyl)methyl]-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
2-{[3-(4-carboxyphenyl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
dimethyl(3-{2-[1-(2-methylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
2-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
2,9-dimethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
2-[1-(2-fluorophenyl)-5-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}piperazine
({5-[1-(1,3-benzothiazole-6-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
6-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{5-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
2-[5-(5-phenoxyfuran-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N3-[2-(3-chlorophenyl)ethyl]-1-cyclohexyl-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S)-N,N-dimethyl-1-(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
5-oxo-N-[2-(pyridin-4-yl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
N-(3-chloro-4-fluorophenyl)-N'-[2-(2-methoxyphenyl)ethyl]propanediamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(1-benzothiophen-5-ylmethyl)-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-tert-butyl-5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazole
2,4-dioxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(4-{[2-(1-hydroxycyclopentyl)ethyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
4-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}benzamide
4-[5-(4-methylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-({1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
2-(4-methyl-3-phenylpiperazine-1-carbonyl)benzene-1,3-diol
N-(1,4-dioxan-2-ylmethyl)-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N,N-dimethyl-2-(4-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)acetamide
2-{1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}ethan-1-ol
2-{9-[2-(2-methoxyphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-4-hydroxy-N,2-dimethylpyrimidine-5-carboxamide
4-(pyridin-4-ylmethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
5-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-1-azabicyclo[3.2.1]octane
N-methyl-2-(methylsulfanyl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
(3-{2-[1-(4-methoxy-3-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-(1H-pyrazol-1-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-oxazepane
N-ethyl-2-{[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amino}pyridine-4-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(morpholin-3-yl)acetyl]piperazin-2-one