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1-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-phenylethane-1,2-dione
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-phenylcyclopropane-1-carboxamide
1-(2,3-dihydro-1H-isoindol-2-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
(1S,6R)-9-[(4-methanesulfonylphenyl)methyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(dimethyl-1,2-oxazol-4-yl)-4-{[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}benzamide
1-(1H-pyrrole-2-carbonyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
N-(4-methoxy-3-propanamidophenyl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
(4aS,8aR)-6-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-chloro-N-(1,2-oxazol-3-ylmethyl)quinoline-2-carboxamide
ethyl 2,4-dimethyl-5-{[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}-1H-pyrrole-3-carboxylate
2-[methyl(pyridin-3-ylmethyl)amino]-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
4,6-dimethyl-1-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
3-(3-methoxyphenyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
1-{4-fluoro-3-[3-(1H-imidazol-1-yl)propyl]phenyl}ethan-1-one
3-[(3-chlorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-(azetidine-1-carbonyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]benzene-1-sulfonamide
4-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
5-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-2-methyl-1,3-benzothiazole
4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
4-fluoro-N-({1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}methyl)benzamide
3-{[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyrimidin-2-one
3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-(piperidin-4-ylmethyl)urea
5-fluoro-1,3-dimethyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl]methanol
2-benzyl-9-[(2R)-3-hydroxy-2-methylpropyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(3-ethylpiperazin-1-yl)-3-oxopropyl]-N-methylbenzene-1-sulfonamide
5-methyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-propyl-1H-pyrazole
(3S,4S)-1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
5-{[(4aS,7aR)-4-cyclobutanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl](methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
7-[(5-ethylfuran-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
N-{1-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl}acetamide
[(5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2,3-dihydro-1H-inden-2-amine
3-{1-[4-(dimethylamino)benzoyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
N-benzyl-1-(cyclohexylmethyl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
N-[2-(pyridin-3-yloxy)ethyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
5-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
2-[methyl({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]ethan-1-ol
3-[5-(2-methoxynaphthalen-1-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
4-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
2-(1H-imidazol-2-yl)-N-methyl-N-[2-(morpholin-4-yl)propyl]benzamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
methyl 4-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidin-1-yl}pentanoate
(3R,4S)-4-cyclopropyl-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-amine