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7-(2,3-dihydro-1H-isoindol-2-ylmethyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-N'-(4-methylphenyl)propanediamide
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(5-fluoropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-(5-methyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]piperidine-1-sulfonamide
7-[(3,4-difluorophenyl)methyl]-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
2-(2-benzylmorpholin-4-yl)-N-(1-methyl-1H-pyrazol-4-yl)acetamide
9-(2-methoxybutanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-chlorophenyl)-4-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
1-cyclohexyl-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(thiophen-2-yl)acetamide
(3aR,6aR)-2-(3,4-dimethylbenzoyl)-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1S)-1-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-3-(methylsulfanyl)propyl]acetamide
1-[1'-(3-fluoropyridin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
8-(2-ethylpyridine-4-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(morpholin-4-yl)benzamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxamide
1-{1'-[2-(4-fluorophenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-{[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[(3-methylquinolin-2-yl)amino]methyl}-1λ6-thiolane-1,1-dione
1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
2-{cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(cyclopropylmethyl)-5-methoxybenzamide
8-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidine
7-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline
4-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
3-{[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
ethyl 4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperazine-1-carboxylate
2-benzyl-8-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3,5-dimethoxybenzamide
(1R,5S,6S)-3-cyclopentyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-(1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)pyridine
6,7-dimethyl-2-{2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}-1H-1,3-benzodiazole
5-(3-fluorophenoxymethyl)-N-(2-oxopyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
methyl({[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
(3S,4S)-1-[(dimethyl-1,3-thiazol-5-yl)sulfonyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-(1-benzyl-1H-pyrazol-3-yl)-2-(4-methyl-1H-imidazol-1-yl)acetamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-(4-phenyl-1H-imidazole-5-carbonyl)piperidine
3-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)-1,2-benzothiazole
N-[(2R,3R)-1'-(2,5-dimethylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-{[3-(3-chlorophenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(2-methylpropyl)piperidin-4-yl]methyl}amine
1-(cyclohexylmethyl)-4-oxo-N-(propan-2-yl)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,4-dihydropyridine-3-carboxamide
1-(3-hydroxypropyl)-4-(4-methoxypyridine-2-carbonyl)-1,4-diazepan-6-ol