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N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-(2-hydroxyacetyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[1-(3,4-dimethoxyphenyl)propyl]-2,6-dimethylpyridine-4-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-5-methyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
1-benzyl-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-2-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-cyclopentyl-2-phenylacetyl)-4-(2-methoxyethyl)-1,4-diazepan-5-one
N-{2-[1-(3,4-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
3-cyclopentyl-5-(1,4-dioxan-2-yl)-1-(3-fluorophenyl)-1H-1,2,4-triazole
(2S,4S)-4-amino-N,N-diethyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
3-methoxy-2-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
3-{1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-N-[furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[2-(4-fluorophenyl)ethyl]propanamide
5-({[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}methyl)-1,2,4-oxadiazole-3-carboxamide
2-ethyl-4-phenyl-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecane
5-(5-cyclopropyl-1,3-oxazol-4-yl)-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
1-[(4aR,8aR)-4a-hydroxy-7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(piperidin-1-yl)ethyl]amine
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
1-{2-[4-(2-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
[2-(diethylamino)ethyl](methyl){[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(5-methylthiophen-2-yl)methyl]amine
1-cyclopropyl-4-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-one
2-cyclopropyl-4-methyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyrimidine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-1,3-benzoxazole
2-ethyl-4-methyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1,3-thiazole-5-carboxamide
(4aS,8aR)-6-(2-methylfuran-3-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-fluoro-3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}benzene-1-sulfonamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
N-(1,3-diphenyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
8-methoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-ethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-[6-hydroxy-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
1-{2-[4-(1H-indol-4-ylmethyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
[(2S)-1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
2-(2-{[2-(2-oxopiperidin-1-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
5-(azocane-1-carbonyl)-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
4-methoxy-2-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
ethyl 3-{5-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}propanoate
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-1-(pyridin-2-yl)piperidine-3-carboxamide
5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-(4-methylphenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
5-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-({5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-[3-(methylsulfamoyl)phenyl]urea