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{2-[(4,6-dimethoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
4,4,4-trifluoro-1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}butan-1-one
2,5-dimethyl-3-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
4-{1-[1-(3-methoxypropyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)piperidin-2-one
6-chloro-N,N-dimethyl-3-({[2-(methylsulfanyl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
1-[2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
2-(3,5-difluorophenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-[2-(5-fluoropentyl)phenyl]-5-methyl-1,3,4-oxadiazole
2,6-dimethoxy-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-3-carboxamide
3-(2-chlorophenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-phenylpropanamide
3-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propane-1,2-diol
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}propan-1-one
N-[1-(6-methoxynaphthalen-2-yl)ethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S,4S)-4-amino-1-[5-(2-chlorophenyl)furan-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
3-(3-hydroxyphenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetamide
1-cyclopentyl-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperazin-2-one
7-(1H-indole-2-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4R)-N,N-diethyl-4-(2-hydroxy-4-methylbenzamido)-1-propanoylpyrrolidine-2-carboxamide
2-(1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
2-methyl-1-[3-(morpholin-4-yl)piperidin-1-yl]-2-phenylpropan-1-one
4-ethyl-1-methyl-3-{[1-(2-propylpyridine-4-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-1-methyl-5-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide
1-(4-sulfamoylphenyl)-3-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethan-1-one
4-{[1-(2-chlorophenyl)ethyl]amino}-1λ4-thian-1-one
2-methyl-4-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(naphthalen-1-yl)-3-{[(1s,4s)-4-hydroxycyclohexyl]formamido}propanamide
N-(3-chloro-2-methylphenyl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{3-[2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propyl}pyridine
3-(2-methoxyethyl)-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxylic acid
8-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-1-(1-{6-[3-(methylsulfanyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
(3aS,6aS)-2-acetyl-5-[(cyclopentylcarbamoyl)carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-chloro-4-({[2-(furan-2-ylmethyl)-3-hydroxypropyl]carbamoyl}amino)-N,N-dimethylbenzamide
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-(2-methoxyphenyl)-1H-pyrazole
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-[(pyridin-2-ylmethyl)amino]pyridine-3-carboxamide
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-ethylpyrimidin-2-amine
[(2S)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
3-methyl-N-[(1-{[2-(methylamino)pyridin-3-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
1-cyclopropyl-4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}pyrrolidin-2-one
3-(oxolan-3-yl)-5-(trimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate