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N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-methanesulfonylacetamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
7-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-methyl-4-{4-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
1-(4-{[(2R,5S)-5-[(1-methyl-1H-indazol-5-yl)methyl]oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(morpholin-4-yl)-3-[2-(pyridin-4-yl)phenoxy]propan-2-ol
N-(4-{1-[(4-sulfamoylphenyl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
4-[(dipropylamino)methyl]-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]benzamide
(2S)-3-(4-hydroxyphenyl)-2-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]propanamide
2-(4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)-N-ethylacetamide
3-[5-(2-methyl-1,3-oxazol-4-yl)-4-phenyl-1H-imidazol-1-yl]butanoic acid
7-fluoro-2-methyl-4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]quinoline
N-(6-phenoxypyridin-3-yl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
3-{[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}phenol
1-(furan-2-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-(1H-imidazol-1-ylmethyl)-1-(4-methylpyrimidin-2-yl)piperidin-4-ol
4-(4-methoxy-3-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N,5-diethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
methyl 1-({[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]carbamoyl}methyl)-1H-pyrazole-3-carboxylate
4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[6-(2-aminoethyl)pyrimidin-4-yl]amino}-1-(2-methoxyphenyl)pyrrolidin-2-one
4-[5-(4-phenyl-1H-imidazol-5-yl)-1,3-thiazol-2-yl]morpholine
3-[2-(3,5-difluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)acetamide
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-methoxypropan-1-one
1-cyclopentyl-4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-{3-[(3-methoxypyrrolidin-1-yl)methyl]phenoxymethyl}pyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
1-[1-(6-chloro-8-methylquinolin-4-yl)piperidin-4-yl]piperidin-4-ol
N-[(5-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-[5-(1-benzofuran-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-ethylpyrrolidin-2-one
N-[(3R,5S)-5-(methylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-(2-hydroxyethyl)-2,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoxaline-6-carboxamide
1-(4-chlorophenyl)-N-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)methyl]cyclopropane-1-carboxamide
1-benzyl-5-(4-methylpiperidine-1-carbonyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-4-methylbenzamide
(2S,4S)-4-amino-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
7-(7-methoxy-4-methylquinolin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[(3R)-pyrrolidin-3-yl]urea
ethyl 1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidine-4-carboxylate
N-cyclohexyl-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-1-yl}propan-1-one
N-({7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
(1R,3S,4S)-3-hydroxy-N-(3-methoxy-2,2-dimethylpropyl)-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carboxamide
N-{[7-(dimethyl-1,3-thiazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
N-benzyl-2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-sulfonamide