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3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yloxy)acetamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N,N-dimethyl-2-{[2-(methylsulfanyl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}adamantane-1-carboxamide
2,2-dimethyl-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]oxane-4-carboxamide
6-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
5-{2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1,4-diazepane
4-fluoro-3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]benzene-1-sulfonamide
1-(3-methoxypyrazin-2-yl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
[(3R,5R)-1-(4-fluoro-2-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-{4-[(4-methyl-1,3-thiazol-2-yl)carbamoyl]phenyl}-1H-imidazole-4-carboxylic acid
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide
4-(4-fluoro-2-hydroxyphenyl)-5,7-dimethoxy-1,2,3,4-tetrahydroquinolin-2-one
methyl 5-(cyclobutylamino)-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[(4-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-N-methyl-N-[1-(pyridin-3-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-1,2-oxazole-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-cyclopentyl-1,2-oxazole-3-carboxamide
N-[2-(methylamino)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
N-[(3S,4R)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
dimethyl[2-(2-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)ethyl]amine
1-(3-methoxybenzoyl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazine
[(2S,4R)-4-(dimethylamino)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N,N-dimethyl-6-{[1-(2-phenylethyl)piperidin-3-yl]amino}pyridine-3-carboxamide
ethyl 1-(cyclopropylmethyl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]acetamide
3-hydroxy-4-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
5-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
(3R,4R)-4-(hydroxymethyl)-1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperidin-3-ol
N-[5-(1H-imidazol-1-yl)pyridin-2-yl]methanesulfonamide
1-(oxane-4-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
methyl 4-({1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)benzoate
6-chloro-N,N-dimethyl-3-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
7-[(4-fluorophenyl)methyl]-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[(4-phenyloxan-4-yl)methyl]urea
2-{1-benzyl-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3,3,3-trifluoropropan-1-one
5-methoxy-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
1-[(4aR,8aR)-6-[2-(2-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-3-(thiophen-2-yl)propan-1-one
ethyl 2-{1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidin-2-yl}acetate
methyl 3-(2,3-dimethylbenzamido)-6-{[(2-ethoxy-2-oxoethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-3,5-dimethylbenzamide
(3aS,7aR)-2-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylphenyl)benzamide