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4-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
1-[(2S,4R)-1-(cyclohexylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)pyridazine-3-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(pyrrolidine-1-carbonyl)piperidine
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(benzyloxy)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
8-methoxy-2-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
1-methyl-4-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[4-fluoro-3-(trifluoromethyl)phenyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-(2-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(3-phenoxypropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(2,5-dimethoxyphenyl)-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
5-cyclopropanecarbonyl-1'-(1H-indole-6-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-(2-{[cyclohexyl(prop-2-yn-1-yl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
N-methyl-5-[(methylsulfanyl)methyl]-N-[2-(oxan-4-yl)ethyl]furan-2-carboxamide
N-[4-({[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
1-(5-chloropyridine-2-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-(2,4-difluorobenzoyl)-3-(3-ethylphenoxy)azetidine
N-[2-(benzyloxy)ethyl]-5-methyl-1,3-oxazole-4-carboxamide
1-(4-acetylphenyl)-3-{[1-(ethoxymethyl)cyclobutyl]methyl}urea
9-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
5-(1H-indol-1-ylmethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
(1S,5R)-3-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
5-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
5-(5-fluoro-1H-indole-2-carbonyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2-methoxyethyl)-N,5-dimethyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
4-hydroxy-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1-(oxolan-2-ylmethyl)urea
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-oxopiperidin-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
2-(3-chlorophenyl)-2-hydroxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[4-(1,4-diazepan-1-ylmethyl)-2,6-dimethoxyphenoxy]propanoic acid
2-(3-methylbutyl)-8-(2-propoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2H-1,3-benzodioxole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-(1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-ethyl-N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]pyrimidine-5-carboxamide
2-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-N-[(2-methoxyphenyl)methyl]formamido]acetic acid
(2E)-N-{[3-methyl-7-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-{3-[4-(1,4-oxazepan-4-yl)piperidin-1-yl]phenyl}pyrrolidin-2-one
5-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
1-methyl-1-[(3-methylpyridin-4-yl)methyl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
2-{2-[(1,4-dithiepan-6-yl)amino]ethyl}-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(cyclohexylmethyl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
5,6-dimethyl-1-{[3-(1,2-oxazinane-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole