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3-[2-(trifluoromethyl)morpholine-4-carbonyl]isoquinoline
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]cycloheptanecarboxamide
1-({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)azetidin-3-ol
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-(1-ethylpiperidin-4-yl)acetamide
2,6,8-trimethyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
8-cyclopropanecarbonyl-2-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3aS,6aS)-2-[(3-chloro-4-propoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-butyl-N-(furan-2-ylmethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[4-(6-methylpyridin-2-yl)-1H-pyrazol-1-yl]acetamide
4-[(3-cyanopiperidin-1-yl)sulfonyl]-N-(2,2-difluoroethyl)benzamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}propanamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(2-methoxyphenyl)methyl]propanamide
(4aS,8aR)-1-(3-aminopropyl)-6-(2,5-dimethylfuran-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[5-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-(3-acetylphenyl)-1-methyl-6-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(pyridin-2-yl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]piperidine-1-carboxamide
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]quinoxaline-5-carboxamide
1-[4-(furan-2-yl)phenyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-amine
1-(3-chlorophenyl)-4-[2-(1H-imidazol-1-yl)acetyl]-5-methylpiperazin-2-one
8-[(2,5-dimethylthiophen-3-yl)sulfonyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-methylphenyl)methyl](prop-2-en-1-yl)amine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(morpholin-4-yl)propyl]acetamide
N-({1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclopropanecarboxamide
1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-propanoylpyrrolidine-2-carboxamide
2-[2-(4-fluorophenoxy)ethyl]-2-azaspiro[4.4]nonan-3-one
N-(2-oxopyrrolidin-3-yl)-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
1-({4-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-3-methoxyphenyl}methyl)-1,4-diazepan-5-one
({4-[2-(dimethylamino)ethoxy]phenyl}methyl)(1H-imidazol-2-ylmethyl)methylamine
3-methyl-4-{1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]piperidin-3-amine
6-(3-chlorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
8-[(2-fluoro-4-methoxyphenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-5-phenylpentan-1-one
(3R,4S)-4-(3-methoxyphenyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-amine
N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-N,1-dimethylpyrrolidin-3-amine
5-{2-[(2-methoxyethyl)amino]ethyl}-1-(2-phenylethyl)pyrrolidin-2-one
4-{[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]methyl}-1H-indole
3-[2-(2,6-difluorophenyl)ethyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
4-(2-fluoro-5-methoxyphenyl)-3-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(1-methoxybutan-2-yl)-3-{methyl[(methylcarbamoyl)methyl]sulfamoyl}benzamide
7-(1H-imidazole-2-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
1-{1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}piperidin-4-amine
4-(4-methyl-1H-imidazole-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-(thiophene-2-sulfonamidomethyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
4,6-dimethyl-1-{3-oxo-3-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propyl}-1,2-dihydropyrimidin-2-one