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1-methyl-6-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,6-dihydropyridazine-3-carboxamide
2-{5-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-imidazole
4-(3-fluorophenoxy)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
4-methoxy-2-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
5-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)pyrazolo[1,5-a]pyrimidin-7-amine
7-methyl-4-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-ethyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-(2-amino-2-methylpropanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
2-[2-(phenylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyridine-3-carboxamide
N-(1-methyl-1H-pyrazol-4-yl)-3-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}benzamide
{3-[(2,4-difluorophenyl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl}methanol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(3-phenylpropyl)piperidine-3-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-4-yl)acetamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(1,2-oxazol-3-ylmethyl)benzamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3,4-difluorophenyl)propanamide
2-(2-fluoro-6-methoxyphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
methyl 1-[(3R,5S)-5-(cycloheptylcarbamoyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(3S,4S)-3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-1-yl]-2,2-dimethylpropan-1-one
1-[(3-methoxyphenyl)methyl]-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N1-(pyridin-3-yl)-N2-(thiolan-3-yl)ethane-1,2-diamine
2-{[4-(2-chlorophenyl)-5-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2S)-2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]-3-(pyridin-4-yl)propanoic acid
4-benzyl-3-ethyl-1-(2-methoxypyridine-3-carbonyl)-1,4-diazepan-5-one
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(furan-2-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-oxoacetamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,4-dimethylbenzamide
1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-phenylpiperazine
{[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amine
2-(2-methoxyphenyl)-N-(1-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)acetamide
3-(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-ethyl-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-phenyl-1H-imidazol-5-yl)pyrimidin-2-amine
1-(1-methyl-1H-pyrrol-2-yl)-2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethane-1,2-dione
3-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyridin-2-ol
1-methyl-N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}-4-oxo-1,4-dihydroquinoline-3-carboxamide
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[(3-methylpyridin-4-yl)methyl]amine
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(thiophene-2-carbonyl)piperazine
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N-cyclopropyl-1-[(1s,4s)-4-[(2E)-3-(thiophen-2-yl)prop-2-enamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
2-(ethylamino)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}pyrimidine-5-carboxamide
5-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-propyl-1H-pyrazole-4-carboxamide
1-[(1R,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-[(3-hydroxypiperidin-1-yl)methyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
3-[2-(2-fluorophenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione