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methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(thiophen-2-ylmethyl)amine
3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3,3-dimethylbutan-1-one
N3-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
2-ethoxy-3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
4-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 1-[(3S,5S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(3-chloro-4-fluorophenyl)-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}propanamide
(3S,4R)-4-(4-fluorophenyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methyl-4-(trifluoromethyl)pyridine
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[6-(dimethylamino)pyrimidin-4-yl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[1-(3-methylbut-2-en-1-yl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-[(2S)-2-hydroxy-3-phenylpropanoyl]-1-(3-methoxyphenyl)piperazin-2-one
(4aS,8aR)-1-propyl-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
methyl 6-[(3,5-dimethylphenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(2-oxopiperidin-1-yl)propanamide
3,5-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]furan-2-carboxamide
1-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-indole-3-carboxamide
1-{3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}azepan-2-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-methanesulfonylpropan-1-one
1-{2-[4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenoxy]ethyl}-1H-imidazole
N-(1,3-benzothiazol-2-yl)-3-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzamide
(2S)-2-[4-(5-ethylfuran-2-yl)-1H-1,2,3-triazol-1-yl]-4-methylpentanamide
2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(2-chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
2-[(butylamino)methyl]-6-fluoroquinolin-4-ol
N-(3-hydroxypropyl)-2,6-dimethyl-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-ethyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-ethyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[(2-methylphenyl)methyl]benzamide
4-(1H-imidazol-1-yl)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]butan-1-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
4-{[5-(2-butyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}azepane
7-[(4-fluorophenyl)methyl]-2-(1H-imidazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(thiophen-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methoxyphenyl)ethan-1-one
5-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]-1,2-dihydropyridin-2-one
2-cyclopentyl-1-{3-[4-(thiomorpholin-4-ylmethyl)phenoxymethyl]piperidin-1-yl}ethan-1-one
(4S,6R)-4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-6-methyl-1,3-diazinane-2-thione
3-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-(4-methoxyphenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]cyclopentane-1-carboxamide
5-(2-ethoxyphenyl)-1,3-benzothiazol-2-amine
4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(3R,4S)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
4-[(1R)-1-(4-chlorophenyl)ethyl]-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-benzyl-9-(5-hydroxypyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one