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N-(butan-2-yl)-N-cyclopentyl-3-(pyrimidin-2-yloxy)benzamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidine
methyl 4-{5-[(4-phenylazepan-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
6-[1-(2-hydroxy-4-methylbenzoyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
2-(4-chlorophenoxy)-1-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
methyl 2-{[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]sulfonyl}benzoate
5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopent-1-ene-1-carboxamide
(3S)-1-ethyl-4-(4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzoyl)-3-methylpiperazin-2-one
4-(azocan-1-yl)-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-2H-1,3-benzodioxole-5-carboxamide
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N-ethylpyrrolidine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
3-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-[2-(thiophen-2-yl)ethyl]urea
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-decahydroisoquinoline
N,N-dimethyl-1-(1-methyl-4-phenylpiperidine-4-carbonyl)azepan-4-amine
N-methyl-N-(1H-pyrazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2-oxopyrrolidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
4-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
2-{[5-(3-cyanophenyl)-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(3-chlorophenyl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
4-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]-4-azatricyclo[4.3.1.13,8]undecan-5-one
N-(3-ethoxy-2-hydroxypropyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
7-acetamido-N-[(5-fluoro-2-methylphenyl)methyl]-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-{1-benzyl-5-[2-(1H-imidazol-2-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
2-(5-{1-[2-(methylsulfanyl)benzoyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
1-methyl-2-(morpholin-4-yl)-N-(thiolan-3-yl)-1H-1,3-benzodiazole-5-carboxamide
4-[1-benzyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
1-(3-chlorophenyl)-4-(2-hydroxy-3-methoxybenzoyl)piperazin-2-one
N-[2-(pyridin-3-yloxy)propyl]-1,2,5-oxadiazole-3-carboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}benzonitrile
1-(2-fluorobenzoyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[2-(2-hydroxyphenoxy)acetyl]-1-(2-methylphenyl)piperazin-2-one
3-(3-fluorophenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-propanamidobenzamide
2-(2H-1,3-benzodioxol-5-yl)-1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)ethan-1-one
N-[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
6-methoxy-2-oxo-N-propyl-N-(thiophen-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl})amine
(1S,4S)-2-(3-chlorophenyl)-5-(quinolin-8-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-N,N-dimethylpyrimidin-2-amine
1-(2-methylpropyl)-4-[1-(oxane-4-carbonyl)pyrrolidin-3-yl]piperidine
5-{[benzyl(methyl)amino]methyl}-N-(4-hydroxybutan-2-yl)-N-methyl-1,2-oxazole-3-carboxamide
6-[methyl(pyridin-2-ylmethyl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide