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N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}propanamide
(3S,9aR)-8-benzoyl-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[4-(4-methoxyphenyl)butan-2-yl]amino}hexan-1-ol
N-[3-(4-methylpiperazin-1-yl)butyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})methylamine
6-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
2-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-{4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
methyl 1-[(3S,5S)-1-(2-ethylbutyl)-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(4aS,8aR)-6-[2-(benzyloxy)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-ethyl-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(1S,5R)-6-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
1-[3-(3-fluorophenyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
4-({4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]furan-2-yl}methyl)morpholine
4-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclopropyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazine-2-carboxamide
4-{1-cyclohexyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-N-methyl-1,3-thiazol-2-amine
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-methylpropyl)pyrimidine
(1-methyl-1H-imidazol-2-yl)({1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-4-yl})methanol
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
methyl 5-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-sulfamoylbenzamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[5-(3,5-dichloro-2-methoxyphenyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-(4-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)propan-1-ol
5-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
3-methyl-7-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
6-[(4-fluoro-3-methoxyphenyl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(dimethylamino)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}pyridine-3-carboxamide
(2S,4R)-4-cyclopentaneamido-N-ethyl-1-(2-phenylethyl)pyrrolidine-2-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-(2-methylpropanoyl)-1,4-diazepan-2-one
ethyl 1-(cyclopropylmethyl)-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
1-[(3S,4R)-1-[4-(dimethylamino)benzoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(2S,4S)-4-{2-[(cyclopropylmethyl)sulfanyl]acetamido}-N-ethyl-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(1S,5R)-6-(2-methylbenzenesulfonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-3-(3,4-dimethoxyphenyl)-1-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
5-(3-methoxyphenyl)-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}furan-2-carboxamide