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(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2,2-dimethyloxan-4-amine
N-(2-hydroxyethyl)-2,4-dimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-2-(2-oxoazepan-1-yl)acetamide
1-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{5-[1-(2-methylbenzoyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
N-cyclohexyl-N-ethyl-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
[(2-chloro-6-fluoro-3-methoxyphenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-pyrazol-4-yl)propan-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2H-1,3-benzodioxol-5-yl)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)propan-1-one
(1R,7S)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
8-{2-[methyl(propan-2-yl)amino]acetyl}-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(propan-2-yl)-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}morpholine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
ethyl 1-ethyl-5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(oxolan-3-yl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H-imidazole
3-(5-fluoro-2-methoxybenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
(1-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(4-methoxyphenyl)-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
{1-[2-({[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)phenyl]piperidin-4-yl}methanol
2-[2-(2-fluorophenyl)ethyl]-4-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3R,4R)-4-{2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-imidazol-1-yl}pyrrolidin-3-ol
1-methanesulfonyl-N-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-amine
2-[(adamantan-1-ylmethyl)({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,6-trimethylquinoline-4-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(dimethyl-1,3-thiazol-2-yl)methyl]benzamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1-hydroxypropan-2-yl)piperidine-4-carboxamide
6-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(morpholine-4-carbonyl)piperidin-1-yl]ethan-1-one
4-{[5-(1-cycloheptyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
(4aS,8aR)-6-(1-benzofuran-2-ylmethyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
4-(furan-2-yl)-2-[5-(propan-2-yl)-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]pyrimidine
N-cyclopentyl-2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoacetamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
2-benzyl-9-(oxolane-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(5-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
3-({1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[(3-methylpyridin-2-yl)methyl]-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-{2-[1-(3-chloro-2-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide