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2-(dimethylamino)-N,4-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(furan-2-yl)propan-1-one
N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methoxy-N-methyl-5-({[3-(morpholin-4-yl)propyl]carbamoyl}amino)benzamide
1-[(2-methylpyrimidin-5-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
3-propyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-amino-3-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{[2-chloro-4-(2,3-dihydro-1,4-benzodioxin-6-yloxy)-6-methoxyphenyl]methyl}pyrrolidine
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
N2,N2-dimethyl-N5-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-(3-chloro-5-fluorobenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-sulfonamide
2-butyl-N-ethyl-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
8-chloro-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]quinoline
6-[3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carboxylic acid
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(1H-1,2,4-triazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
1-[1-(2-methylbenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-(2,3-dihydro-1H-inden-1-yl)ethan-1-one
3-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetamido]-N-tert-butyl-2-methylbenzamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
2-[3-(4-fluorophenoxymethyl)-5-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-methyl-4-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-amine
2-({4-cyclopropyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
5-methyl-4-[1-(pyrimidin-4-yl)piperidin-4-yl]pyrimidine
7-(1-benzothiophen-3-yl)-4-(2,5-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(2-phenylethyl)piperidin-4-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine
1-[2-(2-methoxyphenyl)ethyl]-3-[3-(piperidine-1-carbonyl)phenyl]urea
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidine
[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-chloro-N-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]benzamide
1-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4-(propan-2-yl)piperazine
2-amino-3-ethyl-N-[2-(2-hydroxyethoxy)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
N,5-dimethyl-2-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole-4-carboxamide
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-3,3-dimethylurea
(1R,5S,6R)-3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(morpholin-4-yl)propyl]propanamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
4-(benzylamino)-2-methyl-N-(propan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
2-hydroxy-3-methyl-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
ethyl 1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidine-3-carboxylate
N-[1-(4-chlorophenyl)cyclobutyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide