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4,6-dimethyl-2-oxo-N-[3-(2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2S,4S)-1-methyl-4-[5-(2-methyl-1,3-oxazol-4-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidine-2-carboxylic acid
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-3-methoxybenzoic acid
(3S,4S)-3-hydroxy-4-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-1λ6-thiolane-1,1-dione
6-(3-chloro-5-methoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-[(benzylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
5-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}-2-(methoxymethyl)pyrimidine
1-[(4-chlorophenyl)methyl]-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[(3-hydroxypyrrolidin-1-yl)sulfonyl]-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
{1-[(2E)-2-methylbut-2-en-1-yl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]isoquinoline-5-carboxamide
N-(2-hydroxyethyl)-N-methyl-1-(1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperazin-1-yl}pyrimidine
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
{2-[(2,1,3-benzoxadiazol-5-ylmethyl)[(3-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
N-[4-({6-[(3,5-dimethoxyphenyl)methoxy]-3-oxo-4-(propan-2-yl)-1,4-diazepan-1-yl}methyl)phenyl]acetamide
1'-(4-ethoxybenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-methyl-6-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-1,3-benzothiazol-2-amine
4-[2-(4-fluorophenyl)-3-oxopiperazine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
9-methoxy-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(4-fluorophenoxy)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
(dicyclopropylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
(3R,4R)-N-(9H-fluoren-2-yl)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
2-(5-fluoro-2-methylphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
(2R,6R)-1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(propan-2-yl)pyrimidine
N-[1-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
6-methyl-5-{5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(thian-4-yl)piperazine
3-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(3-hydroxypiperidin-3-yl)methyl]urea
5-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(pyridin-3-yl)propanamide
6-{[benzyl(butyl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
5-acetyl-N-methyl-N-(quinolin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
4-{[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indole
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,4-dimethoxybenzamide
1-{4-[2-(cyclohexylmethyl)morpholin-4-yl]-4-oxobutyl}pyrrolidin-2-one
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-methylpyrimidin-2-amine
2-methyl-6-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
4-({methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(2S,3S)-2-[3-(azetidine-1-carbonyl)benzenesulfonamido]-3-methylpentanamide
N-(1H-indol-5-yl)-4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carboxamide
6-cyclopropyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
3-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-2H-chromen-2-one
(1S,5R)-6-propyl-3-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one