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8-[1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(hydroxymethyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-ol
1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-pyrazol-4-yl)propan-1-one
(1S,5R)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 1-[(3-ethoxy-2-hydroxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-ethyl-2,3-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
N-(1H-indol-4-ylmethyl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
5,6-dimethyl-3-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{5-[6-amino-5-cyano-4-(4-hydroxyphenyl)pyridin-2-yl]thiophen-3-yl}acetic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-[(5-methylfuran-2-yl)methyl]-1,4-diazepane
7-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
3-(2-hydroxyphenyl)-N-(2,2,7-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-pyrazole-5-carboxamide
1-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
N3-[2-(2-aminoethyl)quinazolin-4-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(trifluoromethyl)morpholine
7-(cyclopropylmethyl)-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-4-(4-methylpiperazin-1-yl)-N-(quinolin-5-ylmethyl)benzamide
4-benzyl-3-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(4S)-4-[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-4-acetamidobutanamide
3-methyl-9-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,5,6-trimethylpyrimidin-4-amine
N-[cyclopropyl(4-methoxyphenyl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-[(2S,4S)-1-[(4-chlorophenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(3-methoxyphenyl)amino]butanamide
3-(1-ethyl-1H-imidazol-2-yl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
6-[4-(benzyloxy)-3-methylphenyl]pyrazine-2-carboxylic acid
4-{[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-methanesulfonamido-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}propanamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(methylsulfanyl)propanamide
3-fluoro-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-(3-{[(1,4-dithiepan-6-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
2-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)benzoyl]morpholine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-{2-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
(3S,9aR)-8-benzoyl-3-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}amino)pyridine-4-carboxamide
N-[2-(2-fluorophenyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-(4-propanoylphenoxy)acetamide
4-(1H-imidazol-1-ylmethyl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-ol
ethyl 1-(4-methyl-1,3-oxazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
methyl 4-methyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)benzoate
(1R,2S)-2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(1S,2R)-2-hydroxycyclopentyl]-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(5-methoxy-1H-indazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one