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N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-ethyl-7,8-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-[3-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-3-{5-[2-(methylamino)pyridine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-[(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]morpholine
N-[3-methyl-1-(pyridin-3-yl)butyl]thian-4-amine
[1-(2-chlorophenyl)-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl]dimethylamine
N-cyclopropyl-1-{2-[1-(4-methylbenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(azocan-1-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
2-{4-[(4-ethynylphenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-(methylamino)pyridine-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-4-phenylbutan-1-one
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-[2-(3-fluorophenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N-[(3R,4R)-3-hydroxy-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]pyrazine-2-carboxamide
N,N-dimethyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazine-1-sulfonamide
N-[(1S,2R)-2-aminocyclobutyl]-4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
2-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]ethan-1-ol
(2S,4R)-N-ethyl-4-(3-hydroxypropanamido)-1-(2-methoxy-4-methylbenzoyl)pyrrolidine-2-carboxamide
5-{methyl[1-(thiophen-2-yl)ethyl]amino}-1-[(4-methylphenyl)methyl]azepan-2-one
2-{4-[2-(1H-imidazol-2-yl)benzoyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
N-cyclopropyl-3-[5-(2,5-dimethylfuran-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
methyl 1-{3-[(5-ethylfuran-2-yl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
7-fluoro-N-(thiophen-3-ylmethyl)quinazolin-4-amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]methanol
3-(1H-1,3-benzodiazol-2-yl)-2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}propanoic acid
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-methoxyethoxy)ethan-1-one
1-(4-fluorophenyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepane
4-(3-methylbut-2-en-1-yl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
(4aR,7aS)-1-(3-methylbutanoyl)-4-[3-(1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,9aR)-1-{[3-(thiophen-2-yl)-1H-pyrazol-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
3-[(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
ethyl 4-(2-methoxyethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
2-methyl-6-{2-[(3-methylthiophen-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,3-difluoro-6-methoxybenzoyl)piperidine
6-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
2-ethyl-9-(2-methoxy-5-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carboxamide
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine