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(3S,4R)-3-methoxy-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-4-amine
4-(2-methoxyethoxy)-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
4-chloro-2-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)phenol
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(1R,5R)-N,N-dimethyl-6-(5-propylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(3R,4R)-1-{[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
(4aS,8aR)-6-(cyclopropylmethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
6-methyl-2-(oxolan-2-ylmethyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-(4-aminopyrimidin-2-yl)-4-(cyclopent-3-ene-1-carbonyl)-1,4-diazepane-6-carboxylic acid
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
2-{3-cyclopropyl-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl}-1-ethyl-1H-1,3-benzodiazole
methyl 2-{3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}-4-(methylsulfanyl)butanoate
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
2-[4-(1,4-diazepan-1-ylmethyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
4-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}benzonitrile
N-benzyl-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propanamide
5-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[1-(thian-4-yl)piperidin-4-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]oxy}-3-chloro-N-cyclopentylbenzamide
1-(2-{[(6-methoxyquinolin-8-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
5-(azepane-1-carbonyl)-N-(1-benzothiophen-2-ylmethyl)-1-(butan-2-yl)-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(carbamoylamino)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-N-propylbenzene-1-sulfonamide
(1R,5R)-6-(cyclopropylmethyl)-3-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(5-methylpyrazin-2-yl)methyl]-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
(2S)-2-hydroxy-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
2-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[(3R,4S)-1-cyclopentyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]methanesulfonamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
3-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}propan-1-ol
N-[(1R,3R)-3-aminocyclopentyl]-1-propyl-1H-pyrazole-5-carboxamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-(pyrrolidin-3-yl)acetamide
1-(2-{4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
1-{4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
N-[2-(3-fluorophenyl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
8-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,2-oxazinane
(3S,4S)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
3-benzyl-7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(1R,5R)-6-(5-chlorothiophene-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane