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1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-4-yl)piperazine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
(2S,4R)-4-amino-1-[(4-acetamidophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
{[5-(oxan-2-yl)furan-2-yl]methyl}[(2-phenoxypyridin-3-yl)methyl]amine
1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-ol
1-(4-methyl-1H-pyrrole-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
2-[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-N,N-dimethylacetamide
(1R,9aR)-1-{[(3-phenylpropyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-chloro-1,3-dimethyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1H-pyrazole-4-sulfonamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
(3aS,6aS)-2-(4-chloro-2-fluorobenzoyl)-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(1-methyl-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-(3-hydroxyphenyl)-1-[3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]ethan-1-one
1-cyclopentyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(2-{4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-methyl-6-propyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2-(2-hydroxyethyl)-8-[2-(pyridin-4-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-3-(2-methoxyethyl)-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
5-(2,4-difluorophenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2,6-dimethylpyridine
2-{[1-(3-methylphenyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-[1-(1H-imidazol-2-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N4-(1-benzylpiperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(4-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}phenyl)acetamide
3-[(3R,4S)-1-(3-fluoropyridin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-{1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazol-2-yl}pyridine
3-methyl-4-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
5-(2,3-dihydro-1-benzofuran-5-yl)-3-methylpyridin-2-amine
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[1-(5-chloropyridine-2-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropane-1-carbonitrile
1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-methyl-8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[4.5]decane
9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(methylamino)ethyl]pyridin-2-amine
4-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}piperazin-2-one
1-(2-methoxyacetyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
1-({1-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid