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3-chloro-4-{[1-(1-cyclopropylpropan-2-yl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
2,4-dimethoxy-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2-(pyridin-4-ylmethyl)-9-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-hydroxyphenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-(cyclopropylmethyl)-8-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-amino-4-(4-fluorophenyl)-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
2-(dimethylamino)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
methyl 5-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5-oxopentanoate
2-cyclopentyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
(1S,5R)-N,N-diethyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
dimethyl(2-{2-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidin-1-yl)-5-(trifluoromethyl)pyridine
N-({1-[(3-acetylphenyl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
4-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}morpholine-2-carboxylic acid
2-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-8-fluoroquinoline
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-3-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-(methylsulfanyl)ethan-1-one
N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
5-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-(2-chlorophenyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[(3-methoxyphenyl)methyl]-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(2-hydroxy-4-methoxyphenyl)methyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
N,N-dimethyl-4-({4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)aniline
N-benzyl-5-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)pyrimidin-2-amine
1-[(4-chlorophenyl)methyl]-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperazine
1-[3-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)phenyl]ethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(oxan-4-yl)acetamide
2-methyl-5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}pyrazine
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-(3,5-dimethylphenyl)piperazin-2-one
5-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[3-(3-fluorophenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(2S)-1-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)pyrrolidine-2-carboxamide
1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-4-(oxan-4-yl)piperazine
(3S,4R)-1-(6-aminopyrimidin-4-yl)-3-benzyl-4-methylpiperidin-4-ol
2-[(cyclopentylamino)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
8-chloro-2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]quinoline
2-ethoxy-5-[2-(propylamino)pyrimidin-4-yl]benzoic acid
2-(propan-2-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,3-benzoxazole
5-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
(5S,9aS,9bS)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(2-chloro-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3-fluorophenyl)-4H-1,2,4-triazole
3,4,7-trimethyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
2-[(3-fluorophenyl)methyl]-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]morpholine