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2-{[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzonitrile
4-{3-[(1R)-1-aminoethyl]phenyl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
{2-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}urea
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(trifluoromethyl)benzamide
3-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]-N-phenylpropanamide
N-cyclopropyl-1-[(1s,4s)-4-{[(4-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-{4-[(benzylamino)methyl]-2-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
3-({1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-4-yl}methyl)benzoic acid
4-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]piperazine-2-carboxylic acid
N-(2-hydroxy-3-methoxypropyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}piperidin-2-one
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
methyl N-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}carbamate
2,5-dioxo-6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(4-{2-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-4-chlorophenoxy}piperidin-1-yl)ethan-1-one
3-[3-(4-fluorophenoxy)propyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
ethyl 4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
5-methyl-4-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
2-ethyl-5-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
5-cyclobutanecarbonyl-1'-(6-methylpyridazin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1-propylpiperidin-3-yl)methyl]-4-sulfamoylbenzamide
1-{3-[3-(4-fluorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
2-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}benzoic acid
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-2,3-dihydro-1-benzofuran-5-carboxamide
2-[3-(benzyloxy)propyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(3,4-difluorophenyl)methyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-6-(pyridin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2,3-difluorophenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
2-(pyridin-2-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4,4-difluoro-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-methyl-N-[1-(5-methylpyridin-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(2S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
[(5-methylthiophen-2-yl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
1-(4-chlorobenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxyethan-1-one
5-[4-(3-methoxypropyl)piperidine-1-carbonyl]-1-(2-phenylethyl)piperidin-2-one
1-{[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-N-methylpyridine-3-carboxamide
2-(3-methoxypropyl)-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N,N-diethyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
N-(3-benzylphenyl)-4-(2-propoxyethyl)piperazine-1-carboxamide
4-(2,6-dimethylhept-5-en-1-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol