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4-[(furan-2-ylmethyl)amino]-5-methyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N'-(2-fluoro-5-methylphenyl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]butanediamide
2-methyl-4-(2-methylphenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazine
6-(pyrrolidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
2-[4-oxo-5-(trifluoromethyl)-3,4-dihydroquinazolin-3-yl]acetamide
4-(4-fluoro-2-methoxyphenyl)-6-(methoxymethyl)pyrimidine
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyridine-3-sulfonamide
(1S,5R)-N-(2-ethoxyphenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)propan-1-one
N-cyclopropyl-1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-[(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-ethyl-N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
methyl 3-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}benzoate
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(3,5-dimethoxybenzoyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N4-(1-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
3-{[(5-methylpyrazin-2-yl)methyl]amino}-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
2-ethyl-6-methyl-5-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
5-[4-(2-methoxyethyl)phenoxy]-1-azabicyclo[3.2.1]octane
N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
N-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-phenylmethanesulfonamide
N-[(3S,4R)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-cyclopentyl-2-phenyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
3-[ethyl(pyridin-4-ylmethyl)amino]-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
3-[2-(4-hydroxy-1-methylpiperidin-4-yl)ethyl]-6,8-dimethyl-3,4-dihydroquinazolin-4-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,2-oxazole-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(dimethyl-1,2-oxazol-4-yl)propanamide
8-fluoro-2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
1-[(2-{furo[3,2-c]pyridin-4-yloxy}phenyl)methyl]piperidine
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-benzyl-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-phenoxyacetamide
3-({[(1-benzylpyrrolidin-3-yl)methyl](methyl)amino}methyl)pyridin-2-amine
1-{4-[({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]piperidin-1-yl}ethan-1-one
2-ethyl-8-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-[3-(1,3-oxazol-5-yl)phenyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decane-8-carboxamide
8-fluoro-2-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)methyl]quinolin-4-ol
N-(oxolan-2-ylmethyl)-5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
N-[(2R,3R)-2-methoxy-1'-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
methyl 2-{methyl[1-(thiophen-2-yl)ethyl]carbamoyl}benzoate
2-(2,4-difluorophenyl)-5-(oxolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(1-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol