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[(4aS,8aR)-6-(3,5-dichloro-4-methylbenzoyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-2-phenylethyl]-2-(dimethylamino)-N-methylacetamide
3-(2-ethylbutyl)-8-[(2R)-oxolane-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{3-[6-amino-5-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)pyridin-2-yl]phenyl}acetamide
1-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
6-(methoxymethyl)-2-[3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-(1-benzothiophen-2-ylmethyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-[1-(3-methylbutyl)-1H-pyrazol-5-yl]urea
2-methoxy-N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
methyl[(3-methylpyridin-4-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
2-[3-(1H-imidazol-2-yl)-1H-indol-1-yl]propanoic acid
N-[3-(phenylsulfanyl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(4aR,7aS)-1-acetyl-4-[(3-hydroxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-(2-chloro-4-methoxyphenoxymethyl)-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazole
methyl 2-{1,8-dibenzyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-oxo-4-phenylbutanamide
5-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-2-hydroxybenzoic acid
dimethyl({3-[2-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]propyl})amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,4-dioxane-2-carboxamide
4-chloro-2-[(1E)-3-(3,4-dimethylpiperazin-1-yl)-2-methylprop-1-en-1-yl]phenol
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylpropanamide
2-(2-fluorophenyl)-8-methoxy-5-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-(2-hydroxy-3-methoxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
2-hydroxy-N-({1-[(5-hydroxy-2-methoxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
2-(2,5-dimethylphenoxy)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylpropanamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidine
methyl 3-({1-cyclohexyl-5-[(2-methylpropyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}formamido)propanoate
2-(dimethylamino)-2-(2-fluorophenyl)-N-[1-(hydroxymethyl)cycloheptyl]acetamide
(3R,4S)-4-(3-methoxyphenyl)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-amine
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3S,4R)-1-[2-(1H-imidazol-2-yl)benzoyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
4-{[1-benzyl-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
4-(4-fluorophenyl)-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-oxobutanamide
methyl 3-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)benzoate
5-(2-fluorophenyl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2H-1,3-benzodioxol-5-yloxy)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
1-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[2-(4-propanamidophenoxy)acetyl]piperidine-4-carboxylic acid
1-(2-fluorophenyl)-4-(3-propoxypiperidin-1-yl)piperidine
N-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
N-methyl-4-({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}sulfamoyl)thiophene-2-carboxamide
(1H-imidazol-4-ylmethyl)[(2-methylphenyl)methyl](2-methylpropyl)amine
5-ethyl-1'-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,N-dimethyl-3-[4-(3-methylphenoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
2-(4-methoxyphenyl)-5-[1-(methylsulfanyl)propan-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzoxepine-4-carboxamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(2-methylpropyl)amine