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5-(2-fluorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2,4-triazin-3-amine
3-({4-[(dimethylamino)methyl]-4-hydroxypiperidin-1-yl}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
8-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}quinolin-4-amine
N-[4-(3-methoxyphenyl)phenyl]-1-(1-methylcyclopropanecarbonyl)pyrrolidine-2-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
9-methoxy-7-(4-methylphenyl)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-phenylazetidine-1-carbonyl)-1-(propan-2-yl)piperidine
5-(2-methyloxolane-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[(cyclobutylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-[(5-{[4-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-3,3-dimethylurea
3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-7,8-dimethyl-3,4-dihydroquinazolin-4-one
4-benzyl-3-ethyl-1-(6-ethylpyrimidin-4-yl)-1,4-diazepan-5-one
(4aR,7aS)-1-[(2-ethylphenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2,3-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(1,3-dioxo-2-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
1-[4-(2-methoxyethyl)piperazin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1-methyl-1H-imidazole-4-sulfonamide
4-ethyl-3-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylpyrazine-2-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](2-methoxyethyl)(propan-2-yl)amine
N-methyl-2-(pyridin-2-yl)-N-[2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
methyl 6-(2,3-difluorobenzoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
(4aR,7aS)-1-ethyl-4-[5-(ethylsulfanyl)thiophene-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-{[(1-benzylpiperidin-4-yl)amino]methyl}-4-(pyrimidin-2-yl)phenol
4-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}benzoic acid
N3-(3-{[(4-chlorophenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
1-(pyridin-4-yl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
1-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]azetidine-2-carboxylic acid
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2,3-dimethoxybenzamide
ethyl 1-ethyl-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[2-(thiophen-2-yl)ethyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
(2S,4R)-N-cycloheptyl-1-(3-phenylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(dimethylamino)ethan-1-one
N-({7-fluoro-2-[4-(2-hydroxyethyl)piperazin-1-yl]quinolin-3-yl}methyl)-N-(furan-2-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(1-methoxypropan-2-yl)amino]-5-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
4-hydroxy-N-(3-methoxy-4-methylphenyl)-4-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
N4-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
7-fluoro-N,3-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide