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N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
2-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,7-diazaspiro[4.5]decane
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[3-(2-aminoethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-1H-indole-3-carbonitrile
9-methoxy-7-(3-methoxyphenyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propyl-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
(2,1,3-benzoxadiazol-5-ylmethyl)({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)methylamine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-(furan-3-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(cyclohex-1-en-1-yl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
10-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-(3-methoxyphenyl)-4-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperazin-2-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5-methoxy-1-methyl-1H-indole-2-carboxamide
8-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(1R,3R)-3-aminocyclopentyl]-5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
2-(1H-1,2,3,4-tetrazol-1-yl)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
1-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
6-(4-methanesulfonylphenyl)-2-(morpholin-4-yl)pyrimidin-4-amine
1-methyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-N-{2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]ethyl}methanesulfonamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,6-dimethoxybenzamide
2-[1-(3-methylbutyl)-8-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)propanamide
2-methyl-4-{3-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-(4-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1-methylpiperidin-3-yl)methyl]amine
4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}thiomorpholine
2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-ylmethyl]-4-hydroxyquinoline-6-carboxamide
2-chloro-4-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenol
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-5-methylphenol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](2-methoxyethyl)amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
1-{1-phenyl-2-[2-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}azepane
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-methylurea
(3S,4S)-1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4-cyclopropylpyrrolidine-3-carboxylic acid
methyl 7-oxo-9-(propan-2-yloxy)-3-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-N-(1-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
2-amino-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
4-(2,2-dimethylpropyl)-3-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N,N-dimethyl-2-[(1S,5R)-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(3S,4R)-1-(2-hydroxy-4-methylbenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2,4-dimethylpyrimidine
2-[5-(1-methyl-1H-pyrazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]benzoic acid
1-[(4-methylthiophen-2-yl)sulfonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid