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3-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-2-methyl-1H-indole
(4aS,7aR)-1-(3-hydroxypropanoyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-N-[(4-hydroxyazepan-4-yl)methyl]-5-methoxybenzamide
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-(2-methylphenyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-cyclopropyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(cyclopropylmethyl)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]piperidine-3-carboxylic acid
8-cyclopropanecarbonyl-2-(pyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
2-(2-chlorophenoxy)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
3-({[(2,4-dimethoxyphenyl)methyl]amino}methyl)pyrrolidin-3-ol
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyridin-3-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)acetamide
1-[2-(methylsulfanyl)ethyl]-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
2-methyl-4-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}phenyl)butan-2-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-propanamidobenzamide
ethyl 4-{2-[4-(pyridine-2-amido)-1H-pyrazol-1-yl]acetyl}piperazine-1-carboxylate
10-methoxy-5-[2-(pyrrolidin-3-yl)benzoyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(2-fluoro-4-methylphenyl)-2-{4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}acetamide
3-(pyridin-3-yl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
1-{3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}pyrrolidin-2-one
1-[benzyl(methyl)amino]-3-[5-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-({1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
(3S,4R)-4-(hydroxymethyl)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-3-ol
9-(2-hydroxy-5-methylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
9-(3-methoxypyrazin-2-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(5-chloro-6-methyl-1-benzofuran-3-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
8-[3-(furan-2-yl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(furan-2-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
5-(2-fluorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-cyclobutanecarbonyl-1'-(furan-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,8aR)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-methyl-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine
5-{[methyl({[3-(2-{4-[2-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
methyl 4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-4-oxobutanoate
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(2-hydroxybutyl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
methyl 3-(2-chlorobenzamido)-5-{[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]methyl}benzoate
N-(3-cyano-4-ethoxyphenyl)-4-(5-cyanopyridin-2-yl)piperazine-1-carboxamide
2-methyl-N-{1-[7-(2-methylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
[(3-chlorophenyl)methyl]({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
N-[(3S,4R)-1-(1H-imidazol-4-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
dimethyl(3-{2-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
6-ethyl-N4,5-dimethyl-N4-[(3-methylpyridin-4-yl)methyl]pyrimidine-2,4-diamine
(2S,4S)-4-amino-1-(2,6-dimethoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide