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methyl 5-(2-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclobutyl-N-[(2-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-amine
4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}benzoic acid
N-(3-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)-2-methoxybenzamide
(1S,5R)-3-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-5-(morpholin-4-ylmethyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-cyclohexyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-(benzenesulfonyl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
3-{[(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
3-(1H-1,3-benzodiazol-1-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanamide
2-(2-fluoro-5-methylphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
4-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-[2-(4-chlorophenyl)acetyl]-4-propyl-1,4-diazepan-5-one
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-{[3-(3-methylthiophene-2-carbonyl)piperidine-1-carbonyl]amino}benzoate
2-(morpholin-4-yl)-2-(pyridin-3-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-[(4aR,8aS)-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
4-(3,4-dimethoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
N-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
4-[5-(4-methanesulfonylphenyl)furan-2-carbonyl]morpholine
5-fluoro-1-methyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
4-(1-benzofuran-2-ylmethyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-fluorophenyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrazine-2-carbonyl}morpholine
1-[(3,4-dimethoxypyridin-2-yl)methyl]-5-methylpyrrolidin-2-one
2-chloro-4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-6-methoxyphenol
N-(4-{4-[(5-hydroxyadamantan-2-yl)amino]piperidin-1-yl}phenyl)-2-(4-methoxyphenyl)acetamide
2-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}-1H-1,3-benzodiazole
4-(3-hydroxyazetidine-1-carbonyl)-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
1-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(methylamino)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,3-thiazole-4-carboxamide
7-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[3-(methylsulfanyl)propyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-propylpiperidin-4-amine
1-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2-{3-cyclopentyl-5-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1H-1,3-benzodiazole-2-carboxamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-(3-methylpyridin-4-yl)-4-(5-phenyl-1H-pyrazole-3-carbonyl)-1,4-diazepane
1-(4-aminopiperidin-1-yl)-2-(dimethylamino)-2-(3-methylphenyl)ethan-1-one
6-methyl-2-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-4-(thiomorpholin-4-yl)quinazoline
1-(2,5-dimethoxybenzenesulfonyl)-4-hydroxypiperidine-4-carboxylic acid
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-hydroxy-N-methylbenzamide
ethyl 1-[2-(methylsulfanyl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate